日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Pharmacokinetics, Safety, and Tolerability of the Novel Tetrameric, High-Relaxivity, Macrocyclic Gadolinium-Based Contrast Agent Gadoquatrane in Healthy Adults

新型四聚体高弛豫率大环钆基造影剂Gadoquatrane在健康成人中的药代动力学、安全性和耐受性

Hofmann, Birte Maria; Riecke, Kai; Klein, Stefan; Berse, Matthias; Rottmann, Antje; Sutter, Gabriele; Ebert, Wolfgang

Targeting Plasmodium falciparum IspD in the Methyl-d-erythritol Phosphate Pathway: Urea-Based Compounds with Nanomolar Potency on Target and Low-Micromolar Whole-Cell Activity

针对甲基-d-赤藓糖醇磷酸酯途径中的恶性疟原虫 IspD:具有纳摩尔靶向效力和低微摩尔全细胞活性的尿素基化合物

Daan Willocx, Lorenzo Bizzarri, Alaa Alhayek, Deepika Kannan, Patricia Bravo, Boris Illarionov, Katharina Rox, Jonas Lohse, Markus Fischer, Andreas M Kany, Hannes Hahne, Matthias Rottmann, Matthias Witschel, Audrey Odom John, Mostafa M Hamed, Eleonora Diamanti, Anna K H Hirsch

Regioselective Synthesis of Potential Non-Quinonoid Prodrugs of Plasmodione: Antiparasitic Properties Against Two Hemoglobin-Feeding Parasites and Drug Metabolism Studies

疟原虫酮潜在非醌类前药的区域选择性合成:抗两种以血红蛋白为食的寄生虫的活性及药物代谢研究

Elena Cesar-Rodo ,Baptiste Dupouy ,Cécile Häberli ,Jean-Marc Strub ,David L Williams ,Pascal Mäser ,Matthias Rottmann ,Jennifer Keiser ,Don Antoine Lanfranchi ,Elisabeth Davioud-Charvet

Genetic validation of Pf FKBP35 as an antimalarial drug target

Pf FKBP35 作为抗疟药物靶点的基因验证

Basil T Thommen, Jerzy M Dziekan, Fiona Achcar, Seth Tjia, Armin Passecker, Katarzyna Buczak, Christin Gumpp, Alexander Schmidt, Matthias Rottmann, Christof Grüring, Matthias Marti, Zbynek Bozdech, Nicolas M B Brancucci

Parasite Viability as a Measure of In Vivo Drug Activity in Preclinical and Early Clinical Antimalarial Drug Assessment

寄生虫生存力作为临床前和早期临床抗疟药物评估中体内药物活性的衡量标准

Georges F R Radohery #, Annabelle Walz #, Christin Gumpp, Mohammed H Cherkaoui-Rbati, Nathalie Gobeau, Jeremy Gower, Miles P Davenport, Matthias Rottmann, James S McCarthy, Jörg J Möhrle, Maria Rebelo, Claudia Demarta-Gatsi, David S Khoury

Preclinical Antimalarial Combination Study of M5717, a Plasmodium falciparum Elongation Factor 2 Inhibitor, and Pyronaridine, a Hemozoin Formation Inhibitor

恶性疟原虫延长因子 2 抑制剂 M5717 与疟色素形成抑制剂吡咯萘啶的临床前抗疟联合研究

Matthias Rottmann, Brian Jonat, Christin Gumpp, Satish K Dhingra, Marla J Giddins, Xiaoyan Yin, Lassina Badolo, Beatrice Greco, David A Fidock, Claude Oeuvray, Thomas Spangenberg

Lerisetron Analogues with Antimalarial Properties: Synthesis, Structure-Activity Relationship Studies, and Biological Assessment

具有抗疟特性的雷司琼类似物:合成、构效关系研究和生物学评估

Rudolf Mueller, Virsinha Reddy, Aloysius T Nchinda, Fanuel Mebrahtu, Dale Taylor, Nina Lawrence, Lloyd Tanner, Marine Barnabe, Charles J Eyermann, Bin Zou, Ravinder R Kondreddi, Suresh B Lakshminarayana, Matthias Rottmann, Leslie J Street, Kelly Chibale

The Hyperpolarization-Activated HCN4 Channel is Important for Proper Maintenance of Oscillatory Activity in the Thalamocortical System

超极化激活的 HCN4 通道对于丘脑皮质系统振荡活动的正常维持非常重要

Mehrnoush Zobeiri, Rahul Chaudhary, Anne Blaich, Matthias Rottmann, Stefan Herrmann, Patrick Meuth, Pawan Bista, Tatyana Kanyshkova, Annika Lüttjohann, Venu Narayanan, Petra Hundehege, Sven G Meuth, Maria Novella Romanelli, Francisco J Urbano, Hans-Christian Pape, Thomas Budde, Andreas Ludwig

Polyamidoamine Nanoparticles for the Oral Administration of Antimalarial Drugs

用于口服抗疟药物的聚酰胺胺纳米粒子

Elisabet Martí Coma-Cros, Arnau Biosca, Joana Marques, Laura Carol, Patricia Urbán, Diana Berenguer, Maria Cristina Riera, Michael Delves, Robert E Sinden, Juan José Valle-Delgado, Lefteris Spanos, Inga Siden-Kiamos, Paula Pérez, Krijn Paaijmans, Matthias Rottmann, Amedea Manfredi, Paolo Ferruti, El

Pharmacokinetic-pharmacodynamic analysis of spiroindolone analogs and KAE609 in a murine malaria model

小鼠疟疾模型中螺吲哚酮类似物和 KAE609 的药代动力学-药效学分析

Suresh B Lakshminarayana, Céline Freymond, Christoph Fischli, Jing Yu, Sebastian Weber, Anne Goh, Bryan K S Yeung, Paul C Ho, Véronique Dartois, Thierry T Diagana, Matthias Rottmann, Francesca Blasco