Development of novel alpha 2B adrenergic receptor ligands by using a palladium catalyzed Buchwald Hartwig amination with a brominated benzodiazepine

利用钯催化的Buchwald-Hartwig胺化反应，以溴代苯二氮卓类化合物为原料，开发新型α2B肾上腺素能受体配体。