日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Antibacterial macrocyclic peptides reveal a distinct mode of BamA inhibition

抗菌大环肽揭示了一种独特的BamA抑制模式

Walker, Morgan E; Zhu, Wei; Peterson, Janine H; Wang, Hao; Patteson, Jon; Soriano, Aileen; Zhang, Han; Mayhood, Todd; Hou, Yan; Mesbahi-Vasey, Samaneh; Gu, Meigang; Frost, John; Lu, Jun; Johnston, Jennifer; Hipolito, Christopher; Lin, Songnian; Painter, Ronald E; Klein, Daniel; Walji, Abbas; Weinglass, Adam; Kelly, Terri M; Saldanha, Adrian; Schubert, Jeffrey; Bernstein, Harris D; Walker, Scott S

Pharmacological and structural characterization of vibostolimab, a novel anti-TIGIT blocking antibody for cancer immunotherapy

对新型抗TIGIT阻断抗体vibostolimab进行药理学和结构表征,该抗体可用于癌症免疫治疗。

Thierry O Fischmann ,Daniel Malashock ,Eunseon Ahn ,Hongmei Wang ,Komal Pradhan ,Jeffery Grein ,Srishti Chakravorty ,Soheila Bahmanjah ,David Ban ,Ellen Chien ,Mark Hsieh ,Todd Mayhood ,Jing Yuan ,Janica C Wong ,Maribel Beaumont ,Jeanne Baker ,Mark A McCoy ,Mingmei Cai ,Douglas Wilson ,Wendy Blumenschein ,Sybil M G Williams ,Laurence Fayadat-Dilman ,Wolfgang Seghezzi ,Tanya Keenan ,Jin-Hwan Han

Conserved allosteric inhibitory site on the respiratory syncytial virus and human metapneumovirus RNA-dependent RNA polymerases

呼吸道合胞病毒和人类亚肺病毒 RNA 依赖性 RNA 聚合酶上保守的变构抑制位点

Victoria A Kleiner #, Thierry O Fischmann #, John A Howe, Douglas C Beshore, Michael J Eddins, Yan Hou, Todd Mayhood, Daniel Klein, Debbie D Nahas, Bob J Lucas, He Xi, Edward Murray, Daphne Y Ma, Krista Getty, Rachel Fearns

Discovery and multimerization of cross-reactive single-domain antibodies against SARS-like viruses to enhance potency and address emerging SARS-CoV-2 variants

发现和多聚化针对SARS样病毒的交叉反应性单域抗体,以增强效力并应对新出现的SARS-CoV-2变种

Scott A Hollingsworth # ,Cameron L Noland # ,Karin Vroom ,Anasuya Saha ,Miranda Sam ,Qinshan Gao ,Haihong Zhou ,David U Grandy ,Sujata Singh ,Zhiyun Wen ,Christopher Warren ,Xiaohong Shirley Ma ,Daniel Malashock ,Jennifer Galli ,Gwenny Go ,Michael Eddins ,Todd Mayhood ,Karthik Sathiyamoorthy ,Arthur Fridman ,Fahimeh Raoufi ,Yacob Gomez-Llorente ,Andrea Patridge ,Yinyan Tang ,Shi-Juan Chen ,Marc Bailly ,Chengjie Ji ,Laura J Kingsley ,Alan C Cheng ,Bernhard H Geierstanger ,Daniel M Gorman ,Lan Zhang ,Kalyan Pande

Structure of the insulin receptor-insulin complex by single-particle cryo-EM analysis

通过单粒子低温电子显微镜分析胰岛素受体-胰岛素复合物的结构

Giovanna Scapin, Venkata P Dandey, Zhening Zhang, Winifred Prosise, Alan Hruza, Theresa Kelly, Todd Mayhood, Corey Strickland, Clinton S Potter, Bridget Carragher

Chemical Genetic Analysis and Functional Characterization of Staphylococcal Wall Teichoic Acid 2-Epimerases Reveals Unconventional Antibiotic Drug Targets

葡萄球菌细胞壁磷壁酸2-差向异构酶的化学遗传分析和功能表征揭示了非常规抗生素药物靶点

Mann, Paul A; Müller, Anna; Wolff, Kerstin A; Fischmann, Thierry; Wang, Hao; Reed, Patricia; Hou, Yan; Li, Wenjin; Müller, Christa E; Xiao, Jianying; Murgolo, Nicholas; Sher, Xinwei; Mayhood, Todd; Sheth, Payal R; Mirza, Asra; Labroli, Marc; Xiao, Li; McCoy, Mark; Gill, Charles J; Pinho, Mariana G; Schneider, Tanja; Roemer, Terry

Mechanism of action and epitopes of Clostridium difficile toxin B-neutralizing antibody bezlotoxumab revealed by X-ray crystallography

X射线晶体衍射揭示了艰难梭菌毒素B中和抗体贝洛妥珠单抗的作用机制和表位

Orth, Peter; Xiao, Li; Hernandez, Lorraine D; Reichert, Paul; Sheth, Payal R; Beaumont, Maribel; Yang, Xiaoyu; Murgolo, Nicholas; Ermakov, Grigori; DiNunzio, Edward; Racine, Fred; Karczewski, Jerzy; Secore, Susan; Ingram, Richard N; Mayhood, Todd; Strickland, Corey; Therien, Alex G

Validation, performance under field conditions, and cost-effectiveness of Capillus HIV-1/HIV-2 and determine HIV-1/2 rapid human immunodeficiency virus antibody assays using sequential and parallel testing algorithms in Tanzania

在坦桑尼亚,采用序贯和并行检测算法,对Capillus HIV-1/HIV-2和确定HIV-1/2快速人类免疫缺陷病毒抗体检测方法进行验证、现场性能和成本效益评估。

Mayhood, Meghan K; Afwamba, Isaac A; Odhiambo, Christopher O; Ndanu, Epimack; Thielman, Nathan M; Morrissey, Anne B; Shao, John F; Wells Pence, Brian; Crump, John A