日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Proximity-Induced Rewiring of Oncogenic Kinase Triggers Apoptosis

邻近诱导的致癌激酶重编程触发细胞凋亡

Merz, Manuel L; Shoba, Veronika M; Pergu, Rajaiah; Severance, Zachary C; Munkanatta Godage, Dhanushka N P; Deb, Arghya; Kwok, Hui Si; Singh, Prashant; Singh, Sameek; Allen, Jonathan B; Tian, Wenzhi; Gosavi, Pallavi M; Chaudhary, Santosh K; Anokhina, Viktoriya; Weisberg, Ellen L; Payne, N Connor; He, Yao; Dhaliwal, Rohil; Osadchey, Reilly; Shekhar, Mrinal; Mazitschek, Ralph; Rees, Matthew G; Roth, Jennifer A; Cui, Qiang; Griffin, James D; Liau, Brian B; Choudhary, Amit

The contribution of cyclic imide stereoisomers on cereblon-dependent activity

环状酰亚胺立体异构体对脑蛋白依赖性活性的影响

Amako, Yuka; Ichikawa, Saki; Lloyd, Hannah C; Payne, N Connor; Lin, Zhi; Boghossian, Andrew S; Rees, Matthew G; Ronan, Melissa M; Roth, Jennifer A; Zhu, Qian; Budnik, Bogdan; Mazitschek, Ralph; Woo, Christina M

A method for the detection and enrichment of endogenous cereblon substrates.

一种检测和富集内源性 cereblon 底物的方法

Lloyd Hannah C, Li Yuli, Payne N Connor, Zhao Zhenguang, Xu Wenqing, Kroupova Alena, Zollman David, Long Tengfang, Kabir Farah, Chen Mei, Freeman Rebecca, Feng Ethan Yang, Xi Sarah, Hsu Ya-Chieh, Ciulli Alessio, Mazitschek Ralph, Woo Christina M

Phosphorylation-inducing chimera rewires oncogenic kinase to trigger apoptosis.

磷酸化诱导嵌合体重塑致癌激酶以触发细胞凋亡

Merz Manuel L, Shoba Veronika M, Pergu Rajaiah, Severance Zachary C, Munkanatta Godage Dhanushka N P, Deb Arghya, Kwok Hui Si, Singh Prashant, Singh Sameek, Allen Jonathan B, Tian Wenzhi, Gosavi Pallavi M, Chaudhary Santosh K, Anokhina Viktoriya, Weisberg Ellen L, Payne N Connor, He Yao, Osadchey Reilly, Shekhar Mrinal, Mazitschek Ralph, Rees Matthew G, Roth Jennifer A, Cui Qiang, Griffin James D, Liau Brian B, Choudhary Amit

Inhibiting the Keap1/Nrf2 Protein-Protein Interaction with Protein-Like Polymers

利用类蛋白聚合物抑制Keap1/Nrf2蛋白-蛋白相互作用

Carrow, Kendal P; Hamilton, Haylee L; Hopps, Madeline P; Li, Yang; Qiao, Baofu; Payne, N Connor; Thompson, Matthew P; Zhang, Xiaoyu; Magassa, Assa; Fattah, Mara; Agarwal, Shivangi; Vincent, Michael P; Buyanova, Marina; Bertin, Paul A; Mazitschek, Ralph; Olvera de la Cruz, Monica; Johnson, Delinda A; Johnson, Jeffrey A; Gianneschi, Nathan C

Identification of a Polypeptide Inhibitor of O-GlcNAc Transferase with Picomolar Affinity

鉴定出一种对 O-GlcNAc 转移酶具有皮摩尔级亲和力的多肽抑制剂

Hammel, Forrest A; Payne, N Connor; Marando, Victoria M; Mazitschek, Ralph; Walker, Suzanne

Asymmetric Engagement of Dimeric CRL3 (KBTBD4) by the Molecular Glue UM171 Licenses Degradation of HDAC1/2 Complexes

分子胶UM171与二聚体CRL3(KBTBD4)的不对称结合促进HDAC1/2复合物的降解

Yeo, Megan Jr; Zhang, Olivia; Xie, Xiaowen; Nam, Eunju; Payne, Neil Connor; Gosavi, Pallavi M; Kwok, Hui Si; Iram, Irtiza; Lee, Ceejay; Li, Jiaming; Chen, Nicholas J; Jiang, Hanjie; Wang, Zhipeng A; Lee, Kwangwoon; Mao, Haibin; Harry, Stefan A; Barakat, Idris A; Takahashi, Mariko; Waterbury, Amanda L; Barone, Marco; Mattevi, Andrea; Bar-Peled, Liron; Cole, Philip A; Mazitschek, Ralph; Liau, Brian B; Zheng, Ning

Correction: Prolyl-tRNA synthetase as a novel therapeutic target in multiple myeloma

更正:脯氨酰-tRNA合成酶作为多发性骨髓瘤的新型治疗靶点

Kurata, Keiji; James-Bott, Anna; Tye, Mark A; Yamamoto, Leona; Samur, Mehmet K; Tai, Yu-Tzu; Dunford, James; Johansson, Catrine; Senbabaoglu, Filiz; Philpott, Martin; Palmer, Charlotte; Ramasamy, Karthik; Gooding, Sarah; Smilova, Mihaela; Gaeta, Giorgia; Guo, Manman; Christianson, John C; Payne, N Connor; Singh, Kritika; Karagoz, Kubra; Stokes, Matthew E; Ortiz, Maria; Hagner, Patrick; Thakurta, Anjan; Cribbs, Adam; Mazitschek, Ralph; Hideshima, Teru; Anderson, Kenneth C; Oppermann, Udo

Structural and biochemical characterization establishes a detailed understanding of KEAP1-CUL3 complex assembly.

结构和生化表征建立了对 KEAP1-CUL3 复合物组装的详细了解

Adamson Roslin J, Payne N Connor, Bartual Sergio G, Mazitschek Ralph, Bullock Alex N

A randomized, double-blind, placebo-controlled study of histone deacetylase type 6 inhibition for the treatment of painful diabetic peripheral neuropathy

一项随机、双盲、安慰剂对照研究,旨在评估组蛋白去乙酰化酶6型抑制剂治疗糖尿病周围神经疼痛的疗效。

Michelson, David; Chin, William W; Dworkin, Robert H; Freeman, Roy; Herrmann, David N; Mazitschek, Ralph; Pop-Busui, Rodica; Shaibani, Aziz; Vornov, James; Jones, Melissa; Jarpe, Matthew; Hader, Brittany; Viera, Theresa; Hylan, Michelle; Kachmar, Tim; Jones, Simon