日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Yeast Display Technology Enables Rapid Discovery of Low-Nanomolar Macrocyclic Peptide Inhibitors of Human Angiotensin-Converting Enzyme 2

酵母展示技术可快速发现低纳摩尔级人血管紧张素转化酶2大环肽抑制剂

Romanyuk, Zhanna; Bettin, Giacomo; Brear, Paul; Linciano, Sara; Mazzocato, Ylenia; Bonadies, Simone; Zanotto, Ilaria; Mazzucco, Camilla; Monferone, Alan; Soler, Miguel A; Pasut, Gianfranco; Martin, Sara De; Scarso, Alessandro; Heinis, Christian; Rothenberger, Sylvia; Hyvönen, Marko; Angelini, Alessandro

Screening macrocyclic peptide libraries by yeast display allows control of selection process and affinity ranking.

利用酵母展示技术筛选大环肽库可以控制选择过程和亲和力排序

Linciano Sara, Mazzocato Ylenia, Romanyuk Zhanna, Vascon Filippo, Farrera-Soler Lluc, Will Edward, Xing Yuyu, Chen Shiyu, Kumada Yoichi, Simeoni Marta, Scarso Alessandro, Cendron Laura, Heinis Christian, Angelini Alessandro

Combination of Coevolutionary Information and Supervised Learning Enables Generation of Cyclic Peptide Inhibitors with Enhanced Potency from a Small Data Set

结合共进化信息和监督学习,可以从小数据集中生成具有更高效力的环肽抑制剂。

Mazzocato, Ylenia; Frasson, Nicola; Sample, Matthew; Fregonese, Cristian; Pavan, Angela; Caregnato, Alberto; Simeoni, Marta; Scarso, Alessandro; Cendron, Laura; Šulc, Petr; Angelini, Alessandro