Unhooking the Hook: Optimization of the Aurora A Targeting PROTAC JB170 to CCT400028, an In Vitro Degrader Chemical Probe
解开钩子:优化 Aurora A 靶向 PROTAC JB170 至 CCT400028,一种体外降解化学探针
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.5c03024
O'Hanlon, Jack A; Gutsche, Katrin; Müller, Juliane Elisabeth; Ranjan Prusty, Nihar; Mirza, Amin; Roumeliotis, Theodoros I; Yang, Hengzhang; Stubbs, Mark; Hallett, Stephen T; Eing, Lorenz; McAndrew, Peter Craig; Choudhary, Jyoti Sharma; Le Bihan, Yann-Vaï; Caldwell, John; van Montfort, Rob L M; Workman, Paul; Wolf, Elmar; Newton, Gary K; Evans, Lindsay E