日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A fluorescence-based high throughput assay for the determination of small molecule-human serum albumin protein binding.

一种基于荧光的高通量检测方法,用于测定小分子与人血清白蛋白的结合

McCallum Megan M, Pawlak Alan J, Shadrick William R, Simeonov Anton, Jadhav Ajit, Yasgar Adam, Maloney David J, Arnold Leggy A

Peroxisome proliferation-activated receptor δ agonist GW0742 interacts weakly with multiple nuclear receptors, including the vitamin D receptor.

过氧化物酶体增殖激活受体α激动剂GW0742与多种核受体(包括维生素D受体)相互作用较弱

Nandhikonda Premchendar, Yasgar Adam, Baranowski Athena M, Sidhu Preetpal S, McCallum Megan M, Pawlak Alan J, Teske Kelly, Feleke Belaynesh, Yuan Nina Y, Kevin Chinedum, Bikle Daniel D, Ayers Steven D, Webb Paul, Rai Ganesha, Simeonov Anton, Jadhav Ajit, Maloney David, Arnold Leggy A

Discovery of the first irreversible small molecule inhibitors of the interaction between the vitamin D receptor and coactivators.

发现了维生素 D 受体与辅激活剂相互作用的首个不可逆小分子抑制剂

Nandhikonda Premchendar, Lynt Wen Z, McCallum Megan M, Ara Tahniyath, Baranowski Athena M, Yuan Nina Y, Pearson Dana, Bikle Daniel D, Guy R Kiplin, Arnold Leggy A