日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

TNG260 Is a Small-Molecule CoREST Inhibitor That Sensitizes STK11-Mutant Tumors to Anti-PD-1 Immunotherapy.

TNG260 是一种小分子 CoREST 抑制剂,可使 STK11 突变肿瘤对 PD-1 抗肿瘤免疫疗法敏感。

Ahronian Leanne G, Sahu Soumyadip, Zhang Minjie, Patel Ayushi S, Geng Ke, Bhattacharya Reshmee, Falchook Gerald S, Goldman Jonathan W, Spira Alexander I, Punekar Salman R, Spigel David R, Wang Judy S, Skoulidis Ferdinandos, Stephens Janaye, Meynardie Mary, Powell Jaylen M, Lopez Alfonso, Ranieri Michela, Ploszaj Magdalena A, Tan Yi Jer, Lee Yeuan Ting, Yu Yi, Deng Jiehui, Chen Ting, McCarren Patrick, Tsai Alice, Hussain Suleman S, Doyon Brian, Amemiya Kenjie, Ermolieff Jacques, Shahagadkar Preksha, Das Nikitha M, Flynn Lauren R, Shields Julie A, Danielczyk Laney, McMillan Brian J, Mignault Andre, Meier Samuel R, Wu Hsin-Jung, Guerin David J, Whittington Douglas A, Min Chengyin, Sienczylo Iga, Maxwell John P, DiBenedetto Heather J, Watanabe Hideo, Haines Brian B, Huang Alan, Crystal Adam, Andersen Jannik N, Wu Xinyuan, Wong Kwok-Kin

LIG1 Is a Synthetic Lethal Target in BRCA1 Mutant Cancers.

LIG1 是 BRCA1 突变癌症中的合成致死靶点

Martires Lauren Catherine M, Ahronian Leanne G, Pratt Charlotte B, Das Nikitha M, Zhang Xiaobin, Whittington Douglas A, Zhang Hongxiang, Shen Binzhang, Come Jon, McCarren Patrick, Liu Mu-Sen, Min Chengyin, Feng Tianshu, Jahic Haris, Ali Janid A, Aird Daniel R, Li Fang, Andersen Jannik N, Huang Alan, Mallender William D, Nicholson Hilary E

Allosteric inhibitors of Mycobacterium tuberculosis tryptophan synthase

结核分枝杆菌色氨酸合成酶的变构抑制剂

Michalska, Karolina; Chang, Changsoo; Maltseva, Natalia I; Jedrzejczak, Robert; Robertson, Gregory T; Gusovsky, Fabian; McCarren, Patrick; Schreiber, Stuart L; Nag, Partha P; Joachimiak, Andrzej

An unbiased approach to identify endogenous substrates of "histone" deacetylase 8

一种鉴定“组蛋白”去乙酰化酶 8 内源性底物的无偏方法

Olson, David E; Udeshi, Namrata D; Wolfson, Noah A; Pitcairn, Carol Ann; Sullivan, Eric D; Jaffe, Jacob D; Svinkina, Tanya; Natoli, Ted; Lu, Xiaodong; Paulk, Joshiawa; McCarren, Patrick; Wagner, Florence F; Barker, Doug; Howe, Eleanor; Lazzaro, Fanny; Gale, Jennifer P; Zhang, Yan-Ling; Subramanian, Aravind; Fierke, Carol A; Carr, Steven A; Holson, Edward B

An investigation into pharmaceutically relevant mutagenicity data and the influence on Ames predictive potential

对与药物相关的致突变性数据及其对 Ames 预测潜力的影响进行调查

McCarren, Patrick; Springer, Clayton; Whitehead, Lewis

Nitrosonium-catalyzed decomposition of s-nitrosothiols in solution: a theoretical and experimental study

亚硝酰催化溶液中S-亚硝基硫醇的分解:理论与实验研究

Zhao, Yi-Lei; McCarren, Patrick R; Houk, K N; Choi, Bo Yoon; Toone, Eric J