日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Structural and dynamic insights into agonist recognition and function of the thromboxane A(2) receptor

血栓素A2受体激动剂识别和功能的结构和动力学研究

Krawinski, Pawel; Matzov, Donna; Ryder, Aoife; Lal, Kanhaya; Karlov, Dmitry S; Chalhoub, Georges; Mulvaney, Eamon P; Kinsella, B Therese; McCormick, Peter J; Caffrey, Martin; Tikhonova, Irina G; Shalev-Benami, Moran

A network-based atlas of human skeletal muscle aging

基于网络的人类骨骼肌衰老图谱

Stokes, Tanner; Lim, Changhyun; Ali, Muhammad; Mcleod, Jonathan C; Gisby, Jack; Mariniello, Katia; Crossland, Hannah; Sharif, Jalil-Ahmad; Deane, Colleen; Moseley, Thomas C; Ismail, Nasim M; Lixandrao, M E; Volmar, C H; McCormick, Peter J; Brogan, Robert J; Whiteford, James; Roschel, H; Phillips, Stuart M; Gallagher, Iain J; Slabaugh, Gregory; Phillips, Bethan E; Kraus, William E; Atherton, Philip J; Chapple, J Paul; Timmons, James A

MRAP2 modifies the signaling and oligomerization state of the melanocortin-4 receptor.

MRAP2 改变黑皮质素-4 受体的信号传导和寡聚化状态

Sohail Iqra, Laurin Suli-Anne, Kleinau Gunnar, Chunilal Vidicha, Morton Andrew, Brenlla Alfonso, Kagiali Zeynep Cansu Uretmen, Blouin Marie-José, Tello Javier A, Beck-Sickinger Annette G, Lohse Martin J, Scheerer Patrick, Bouvier Michel, McCormick Peter, Annibale Paolo, Biebermann Heike

Multiomics reveal key inflammatory drivers of severe obesity: IL4R, LILRA5, and OSM

多组学揭示重度肥胖的关键炎症驱动因素:IL4R、LILRA5 和 OSM

Chen, Hung-Hsin; Highland, Heather M; Frankel, Elizabeth G; Scartozzi, Alyssa C; Zhang, Xinruo; Roshani, Rashedeh; Sharma, Priya; Kar, Asha; Buchanan, Victoria L; Polikowsky, Hannah G; Petty, Lauren E; Seo, Jungkyun; Anwar, Mohammad Yaser; Kim, Daeeun; Graff, Mariaelisa; Young, Kristin L; Zhu, Wanying; Karastergiou, Kalypso; Shaw, Douglas M; Justice, Anne E; Fernández-Rhodes, Lindsay; Krishnan, Mohanraj; Gutierrez, Absalon; McCormick, Peter J; Aguilar-Salinas, Carlos A; Tusié-Luna, Maria Teresa; Muñoz-Hernandez, Linda Liliana; Herrera-Hernandez, Miguel; Lee, Miryoung; Gamazon, Eric R; Cox, Nancy J; Pajukanta, Päivi; Fried, Susan K; Gordon-Larsen, Penny; Shah, Ravi V; Fisher-Hoch, Susan P; McCormick, Joseph B; North, Kari E; Below, Jennifer E

MACHINE LEARNING-AIDED EXPLORATION OF PHARMACOTHERAPY TO OVERCOME INAPPROPRIATE MULTIPLE MEDICATION AND IMPROVE MOTOR FUNCTION IN THE ELDERLY

利用机器学习辅助探索药物治疗方案,以克服不恰当的多重用药问题并改善老年人的运动功能

Baker, Jillian G; Sloan, Erica K; Pfleger, Kevin D G; McCormick, Peter J; Salmerón, Cristina; Insel, Paul A; Factor, *Sedric John; Ly-Uson, Josefina; Aligam, Katrina Joy; Gelvezon, Marie Angelique; Shigetome, *Keiichi; Oniki, Kentaro; Takata, Keiji; Tateyama, Yuki; Yasuda, Hiroki; Yokota, Miu; Yamauchi, Sae; Yasui-Furukori, Norio; Yamada, Kazunori D; Saruwatari, Junji

Identification of a Cannabinoid Receptor 2 Allosteric Site Using Computational Modeling and Pharmacological Analysis.

利用计算建模和药理学分析鉴定大麻素受体 2 变构位点

Farooq Zara, Delre Pietro, Iliadis Stylianos, Mangiatordi Giuseppe Felice, Contino Marialessandra, Howell Lesley A, McCormick Peter J

Flipping the GPCR Switch: Structure-Based Development of Selective Cannabinoid Receptor 2 Inverse Agonists

翻转GPCR开关:基于结构的选择性大麻素受体2反向激动剂的开发

Kosar, Miroslav; Sarott, Roman C; Sykes, David A; Viray, Alexander E G; Vitale, Rosa Maria; Tomašević, Nataša; Li, Xiaoting; Ganzoni, Rudolf L Z; Kicin, Bilal; Reichert, Lisa; Patej, Kacper J; Gómez-Bouzó, Uxía; Guba, Wolfgang; McCormick, Peter J; Hua, Tian; Gruber, Christian W; Veprintsev, Dmitry B; Frank, James A; Grether, Uwe; Carreira, Erick M

Correction to: A(1)R-A(2A)R heteromers coupled to G(s) and G(i/0) proteins modulate GABA transport into astrocytes

更正:A(1)RA(2A)R异聚体与G(s)和G(i/0)蛋白偶联,调节GABA向星形胶质细胞的转运

Cristóvão-Ferreira, Sofia; Navarro, Gemma; Brugarolas, Marc; Pérez-Capote, Kamil; Vaz, Sandra H; Fattorini, Giorgia; Conti, Fiorenzo; Lluis, Carmen; Ribeiro, Joaquim A; McCormick, Peter J; Casadó, Vicent; Franco, Rafael; Sebastião, Ana M

Wnt signalling in the articular cartilage: A matter of balance

关节软骨中的Wnt信号通路:一种平衡机制

Gill, Amandeep Kaur; McCormick, Peter J; Sochart, David; Nalesso, Giovanna

Detection of cannabinoid receptor type 2 in native cells and zebrafish with a highly potent, cell-permeable fluorescent probe

利用高效、细胞渗透性荧光探针检测天然细胞和斑马鱼中的大麻素受体2型

Gazzi, Thais; Brennecke, Benjamin; Atz, Kenneth; Korn, Claudia; Sykes, David; Forn-Cuni, Gabriel; Pfaff, Patrick; Sarott, Roman C; Westphal, Matthias V; Mostinski, Yelena; Mach, Leonard; Wasinska-Kalwa, Malgorzata; Weise, Marie; Hoare, Bradley L; Miljuš, Tamara; Mexi, Maira; Roth, Nicolas; Koers, Eline J; Guba, Wolfgang; Alker, André; Rufer, Arne C; Kusznir, Eric A; Huber, Sylwia; Raposo, Catarina; Zirwes, Elisabeth A; Osterwald, Anja; Pavlovic, Anto; Moes, Svenja; Beck, Jennifer; Nettekoven, Matthias; Benito-Cuesta, Irene; Grande, Teresa; Drawnel, Faye; Widmer, Gabriella; Holzer, Daniela; van der Wel, Tom; Mandhair, Harpreet; Honer, Michael; Fingerle, Jürgen; Scheffel, Jörg; Broichhagen, Johannes; Gawrisch, Klaus; Romero, Julián; Hillard, Cecilia J; Varga, Zoltan V; van der Stelt, Mario; Pacher, Pal; Gertsch, Jürg; Ullmer, Christoph; McCormick, Peter J; Oddi, Sergio; Spaink, Herman P; Maccarrone, Mauro; Veprintsev, Dmitry B; Carreira, Erick M; Grether, Uwe; Nazaré, Marc