日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Biased Signaling in Psychedelic Action

迷幻剂作用中的偏向信号

Wacker, Daniel; McCorvy, John D

The psychoplastogen tabernanthalog induces neuroplasticity without proximate immediate early gene activation.

精神可塑性物质tabernanthalog可诱导神经可塑性,而无需立即激活早期基因

Aarrestad Isak K, Cameron Lindsay P, Fenton Ethan M, Casey Austen B, Rijsketic Daniel R, Patel Seona D, Sambyal Rohini, Johnson Shane B, Ly Calvin, Viswanathan Jayashri, Barragan Eden V, Lozano Stephanie A, Seban Nicolas, Hu Hongru, Powell Noel A, Chytil Milan, Meyer Retsina, Rose David, Hempel Chris, Olson Eric, Hansen Hanne D, Madsen Clara A, Knudsen Gitte M, Redd Chase, Wheeler Damian G, Guanzon Nathaniel, Muir Jessie, Hennessey Joseph J, Quon Gerald, McCorvy John D, Gandhi Sunil P, Rasmussen Kurt, Liston Conor, Gray John A, Heifets Boris D, Nord Alex S, Kim Christina K, Olson David E

The ABCs of psychedelics: a preclinical roadmap for drug discovery

迷幻药入门:药物发现的临床前路线图

Kwan, Alex C; Mantsch, John R; McCorvy, John D

A Novel Class of Complement 3a Receptor Agonists and Antagonists Derived from the TLQP-21 Peptide

一类源自TLQP-21肽的新型补体3a受体激动剂和拮抗剂

Rodriguez, Pedro; Pallais, Jean Pierre; He, Rongjun; Razzoli, Maria; McKee, John L; Bock, Hailey A; McCorvy, John D; Sham, Yuk Y; DiMarchi, Richard; Bartolomucci, Alessandro

Next-Generation MDMA Analogue SDMA: Pharmacological and Metabolic Insights

下一代MDMA类似物SDMA:药理学和代谢学见解

Kastner, Nina; Nadal-Gratacós, Núria; Hemmer, Selina; Alves da Silva, Leticia; McKee, John L; Hell, Tamara; Cicalese, Giulia; Holy, Marion; Kooti, Fatemeh; Jäntsch, Kathrin; Baron, Ricarda; Shacham, Naomi; Cuccurazzu, Bruna; Halberstadt, Adam L; McCorvy, John D; Stockner, Thomas; Meyer, Markus R; López-Arnau, Raúl; Grill, Matthias; Sitte, Harald H

Serotonin 5-HT(2C) Receptor Signaling Analysis Reveals Psychedelic Biased Agonism

血清素 5-HT(2C) 受体信号分析揭示迷幻剂偏向性激动作用

Bonniwell, Emma M; Alabdali, Rana; Hennessey, Joseph J; McKee, John L; Cavalco, Natalie G; Lammers, Josie C; Moore, Ethan J; Franchini, Luca; Orlandi, Cesare; McCorvy, John D

Assessing the Potential Cardiovascular Risk of Microdosing the Psychedelic LSD in Mice

评估小鼠微剂量服用迷幻药LSD的潜在心血管风险

Effinger, Devin P; Schalk, Serena S; King, Jillian L; Wallingford, Janae R; O'Connell, Caden K; Calderon, Joselynn R; Kopecky, Benjamin J; McCorvy, John D; Thompson, Scott M

Structural basis for selectivity and antagonism in extracellular GPCR-nanobodies

细胞外GPCR纳米抗体选择性和拮抗作用的结构基础

Roman R Schlimgen ,Francis C Peterson ,Raimond Heukers ,Martine J Smit ,John D McCorvy ,Brian F Volkman

Psilocybin analog 4-OH-DiPT enhances fear extinction and GABAergic inhibition of principal neurons in the basolateral amygdala

裸盖菇素类似物 4-OH-DiPT 可增强恐惧消退和基底外侧杏仁核主要神经元的 GABA 能抑制

Kelly, Thomas J; Bonniwell, Emma M; Mu, Lianwei; Liu, Xiaojie; Hu, Ying; Friedman, Vladislav; Yu, Hao; Su, Wantang; McCorvy, John D; Liu, Qing-Song

Potent and Selective Human 5-HT(2B) Serotonin Receptor Antagonists: 4'-Cyano-(N)-methanocarba-adenosines by Synthetic Serendipity

合成意外发现的高效选择性人5-HT(2B)血清素受体拮抗剂:4'-氰基-(N)-甲氧基碳酰胺腺苷

Tosh, Dilip K; Pavan, Matteo; Clark, Allison A; Lammers, Josie; Villano, Serafina; Marri, Silvia; Sgambellone, Silvia; Choi, Suebin; Lee, Jihyun; Ivancich, Marko S; Bock, Hailey A; Campbell, Ryan G; Lewicki, Sarah A; Levitan, Ian M; Chen, Eric; Liu, Naili; Demby, Tamar; Gavrilova, Oksana; Gao, Zhan-Guo; Lucarini, Laura; McCorvy, John D; Jacobson, Kenneth A