Discovery of a benzo[e]pyrimido-[5,4-b][1,4]diazepin-6(11H)-one as a Potent and Selective Inhibitor of Big MAP Kinase 1
发现苯并[e]嘧啶并-[5,4-b][1,4]二氮卓-6(11H)-酮作为 Big MAP 激酶 1 的强效选择性抑制剂
期刊:ACS Medicinal Chemistry Letters
影响因子:3.5
doi:10.1021/ml100304b
Xianming Deng, Qingkai Yang, Nicholas Kwiatkowski, Taebo Sim, Ultan McDermott, Jeffrey E Settleman, Jiing-Dwan Lee, Nathanael S Gray