日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of BMS-986365, a First-in-Class Dual Androgen Receptor Ligand-Directed Degrader and Antagonist, for the Treatment of Advanced Prostate Cancer.

发现 BMS-986365,一种首创的双重雄激素受体配体导向降解剂和拮抗剂,用于治疗晚期前列腺癌。

Nayak Surendra, Norris John D, Ammirante Massimo, Rychak Emily, Wardell Suzanne E, Liao Debbie, Toyama Brandon, Kandimalla Raju, Christoforou Andy, Tsuji Toshiya, Liu Ken, Tran Minerva, Meiring Joseph, Reiss Samantha, Piccotti Joseph R, Baughman Joshua M, Fontanillo Celia, Khater Marwa, Mortensen Deborah S, Cathers Brian, Bence Neil, Pierce Daniel W, Plantevin-Krenitsky Veronique, Rathkopf Dana, Hansen Joshua D, Hamann Lawrence G, Narla Rama Krishna, Arora Vivek K, McDonnell Donald P, Rolfe Mark, Xu Shuichan

Regulation of the immune CD155-CD226-TIGIT axis by cyclin D-CDK4/6

细胞周期蛋白D-CDK4/6对免疫CD155-CD226-TIGIT轴的调控

Fassl, Anne; Palacios Espinoza, Miriam; Butter, Deborah; Kolodziejczyk, Aleksandra; Seehawer, Marco; Hill, Charlotte; Ning, Xiaohan; Branigan, Timothy B; Peñailillo, Johany; Saengboonmee, Charupong; Jadhav, Heta; Charbonnier, Louis-Marie; Waks, Adrienne G; Strawser, Corinne; McDonnell, Donald P; Shapiro, Geoffrey I; Tolaney, Sara M; Polyak, Kornelia; Sammons, Sarah; Wucherpfennig, Kai W; Sicinski, Piotr

Targeting the ERα DBD-LBD Interface with Mitoxantrone Disrupts Receptor Function through Proteasomal Degradation.

利用米托蒽醌靶向 ERα DBD-LBD 界面,通过蛋白酶体降解破坏受体功能。

Wang Han, Luo Yuxuan, Artham Sandeep, Wang Qianqian, Peng Yi, Yun Zixi, Li Xinyue, Wu Chen, Liu Zhenghao, Weber-Bonk Kristen L, Pai Chun-Peng, Cao Yuan, Yue Jiangan, Park Sunghee, Keri Ruth A, Geng Lisheng, McDonnell Donald P, Kao Hung-Ying, Yang Sichun

The Selective Estrogen Receptor Degrader ZN-c5 Has Broad Antitumor Activity in Wild-Type and Mutant ER-Positive Breast Cancer Models.

选择性雌激素受体降解剂 ZN-c5 在野生型和突变型 ER 阳性乳腺癌模型中具有广泛的抗肿瘤活性。

Ma Jianhui, Hegde Sayee, Sergeeva Masha, Chakraborty Binita, Wardell Suzanne E, McDonnell Donald P, Huang Peter Q, Bunker Kevin D, Doñate Fernando, Lackner Mark R, Samatar Ahmed A

Bert W. O’Malley (1936–2025): A great scientist, mentor, and proud Irishman

伯特·W·奥马利(1936–2025):一位伟大的科学家、导师和骄傲的爱尔兰人

Eroume À Egom, Emmanuel; Shiwani, Haaris A; Nouthe, Brice; McDonnell, Donald P

Targeting androgen receptor signaling to enhance cancer immunotherapy

靶向雄激素受体信号通路以增强癌症免疫疗法

Bader, David A; Chakraborty, Binita; McDonnell, Donald P; Hirschey, Matthew D

ESRRA (estrogen related receptor, alpha) induces ribosomal protein RPLP1-mediated adaptive hepatic translation during prolonged starvation.

ESRRA(雌激素相关受体α)在长期饥饿期间诱导核糖体蛋白RPLP1介导的适应性肝脏翻译

Tripathi Madhulika, Gauthier Karine, Sandireddy Reddemma, Zhou Jin, Gupta Priyanka, Sakthivel Suganya, Jiemin Nah, Arul Kabilesh, Tikno Keziah, Park Sung-Hee, Wu Yajun, Wang Lijin, Bay Boon-Huat, Ho Lena, Giguere Vincent, Ghosh Sujoy, McDonnell Donald P, Yen Paul M, Singh Brijesh K

The Impact of Circulating Tumor Cell HOXB13 RNA Detection in Men with Metastatic Castration-Resistant Prostate Cancer (mCRPC) Treated with Abiraterone or Enzalutamide

循环肿瘤细胞 HOXB13 RNA 检测对接受阿比特龙或恩扎卢胺治疗的转移性去势抵抗性前列腺癌 (mCRPC) 患者的影响

Halabi, Susan; Guo, Siyuan; Park, Joseph J; Nanus, David M; George, Daniel J; Antonarakis, Emmanuel S; Danila, Daniel Costin; Szmulewitz, Russell Zelig; McDonnell, Donald P; Norris, John D; Lu, Changxue; Luo, Jun; Armstrong, Andrew J

Estrogen receptor-related receptor (Esrra) induces ribosomal protein Rplp1-mediated adaptive hepatic translation during prolonged starvation

雌激素受体相关受体(Esrra)在长期饥饿期间诱导核糖体蛋白Rplp1介导的适应性肝脏翻译

Tripathi, Madhulika; Gauthier, Karine; Sandireddy, Reddemma; Zhou, Jin; Gupta, Priyanka; Sakthivel, Suganya; Jiemin, Nah; Arul, Kabilesh; Tikno, Keziah; Park, Sung-Hee; Wang, Lijin; Ho, Lena; Giguere, Vincent; Ghosh, Sujoy; McDonnell, Donald P; Yen, Paul M; Singh, Brijesh K

Eosinophilia in cancer and its regulation by sex hormones

癌症中的嗜酸性粒细胞增多症及其受性激素的调节

Artham, Sandeep; Chang, Ching-Yi; McDonnell, Donald P