日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Putative α7-selective ligands interact with α9-containing nicotinic acetylcholine receptors and modulate immune functions of human mononuclear phagocytes

推测的α7选择性配体与含有α9亚基的尼古丁乙酰胆碱受体相互作用,并调节人类单核吞噬细胞的免疫功能。

Mobasher, Mona; Hone, Arik J; Pilzecker, Malin; Bozic, Daria; Hecker, Andreas; McIntosh, J Michael; Kirschner, Karl N; Grau, Veronika; Papke, Roger L; Andleeb, Hina; Richter, Katrin

Hippocampal Metabolomics Reveal the Mechanism of α-Conotoxin [S9K]TxID Attenuating Nicotine Addiction

海马代谢组学揭示α-芋螺毒素[S9K]TxID减轻尼古丁成瘾的机制

Wang, Meiting; Xu, Weifeng; Wang, Huanbai; Cui, Cheng; He, Rongyan; Li, Xiaodan; Yu, Jinpeng; McIntosh, J Michael; Zhangsun, Dongting; Luo, Sulan

Shape-shifting conotoxins reveal divergent pore-targeting mechanisms in nicotinic receptors

形态变化的芋螺毒素揭示了尼古丁受体中不同的孔道靶向机制

Bhattacharjee, Biddut; Noviello, Colleen M; Rahman, Md Mahfuzur; Mayer, John P; Gajewiak, Joanna; McIntosh, J Michael; Hibbs, Ryan E; Stowell, Michael H B

Structural similarities reveal an expansive conotoxin family with a two-finger toxin fold

结构相似性揭示了一个庞大的芋螺毒素家族,其具有双指毒素折叠结构。

Khilji, Muhammad Saad; Hackney, Celeste M; Koch, Thomas L; Hone, Arik J; Rogalski, Aymeric; Watkins, Maren; Tun, Jortan; McIntosh, J Michael; Olivera, Baldomero; Safavi-Hemami, Helena; Teilum, Kaare; Ellgaard, Lars

An N-Terminally Elongated Peptide From Conus rolani Defines a New Class of Ribbon α-Conotoxins Targeting Muscle nAChRs

来自罗兰芋螺的N端延长肽定义了一类靶向肌肉nAChR的新型带状α-芋螺毒素

Giglio, Matías L; Flórez-Salcedo, Paula; Azam, Layla; Watkins, Maren; Koch, Thomas Lund; Basgall-De la Rosa, Erianna; Douglass, Adam D; McIntosh, J Michael; Olivera, Baldomero M; Gajewiak, Joanna

Human α10 nicotinic acetylcholine receptor subunits assemble to form functional receptors

人类α10尼古丁乙酰胆碱受体亚基组装形成功能性受体

Tekarli, Bassel; Azam, Layla; Hone, Arik J; McIntosh, J Michael

Stereoisomers of Chiral Methyl-Substituted Symmetric and Asymmetric Aryl Piperazinium Compounds Exhibit Distinct Selectivity for α9 and α7 Nicotinic Acetylcholine Receptors.

手性甲基取代的对称和不对称芳基哌嗪化合物的立体异构体对α9和α7尼古丁乙酰胆碱受体表现出不同的选择性

Andleeb Hina, Papke Roger L, Richter Katrin, Grau Veronika, Hone Arik J, Kerr Andrew, McIntosh J Michael, Stokes Clare, Thakur Ganesh A

Conotoxins Targeting Voltage-Gated Sodium Ion Channels

靶向电压门控钠离子通道的芋螺毒素

Pei, Shengrong; Wang, Nan; Mei, Zaoli; Zhangsun, Dongting; Craik, David J; McIntosh, J Michael; Zhu, Xiaopeng; Luo, Sulan

Design, Synthesis, and Structure-Activity Relationships of Novel Peptide Derivatives of the Severe Acute Respiratory Syndrome-Coronavirus-2 Spike-Protein that Potently Inhibit Nicotinic Acetylcholine Receptors

强效抑制尼古丁乙酰胆碱受体的严重急性呼吸综合征冠状病毒2刺突蛋白新型肽衍生物的设计、合成及构效关系研究

Hone, Arik J; Santiago, Ulises; Harvey, Peta J; Tekarli, Bassel; Gajewiak, Joanna; Craik, David J; Camacho, Carlos J; McIntosh, J Michael

αO-Conotoxin GeXIVA[1,2] Reduced Neuropathic Pain and Changed Gene Expression in Chronic Oxaliplatin-Induced Neuropathy Mice Model

αO-芋螺毒素GeXIVA[1,2]可减轻慢性奥沙利铂诱导神经病变小鼠模型中的神经性疼痛并改变基因表达

Wang, Huanbai; Li, Xiaodan; Qiao, Yamin; Wang, Meiting; Wang, Wen; McIntosh, J Michael; Zhangsun, Dongting; Luo, Sulan