日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of small molecule inhibitors of PPM1D using an integrated drug discovery platform.

利用综合药物发现平台鉴定PPM1D小分子抑制剂

Shaw Subrata, Jiang Wei, Rush Jason, Dumont Nancy, Kim John, Singh Ritu, Skepner Adam, Khodier Carol, Raffier Cerise, Murphy Zachary, Yan Ni, Schluter Cameron, Yu Xiao, Szuchnicki Mateusz, Sathappa Murugappan, Kahn Josephine, Sperling Adam S, Wagner Florence, McKinney David C, Gould Alexandra E, Garvie Colin W, Miller Peter G

Targeting NEDD9-SH3 with a Covalent Peptide Controls Endothelial Phenotype.

利用共价肽靶向NEDD9-SH3可控制内皮细胞表型

Samokhin Andriy O, Seo Hyuk-Soo, Leed Alison, Hajian Behnoush, Bird Gregory H, McKinney David C, Saha Progyaparamita, Daum Jacqueline, Moroco Jamie A, Yehl Jenna, Kornfilt David, Szczeniowski Anna, Petrunak Elyse, Horner Steven, Kalin Jay H, Leymarie Nancy, Kaushik Virendar K, Walensky Loren D, Cole Philip A, Oldham William M, Steinhauser Matthew L, Dhe-Paganon Sirano, Maron Bradley A

Structural Insights Lead to a Negamycin Analogue with Improved Antimicrobial Activity against Gram-Negative Pathogens

结构解析揭示了一种对革兰氏阴性病原体具有更强抗菌活性的奈加霉素类似物

McKinney, David C; Basarab, Gregory S; Cocozaki, Alexis I; Foulk, Melinda A; Miller, Matthew D; Ruvinsky, Anatoly M; Scott, Clay W; Thakur, Kumar; Zhao, Liang; Buurman, Ed T; Narayan, Sridhar