日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

2-Aminomethylene-5-sulfonylthiazole Inhibitors of Lysyl Oxidase (LOX) and LOXL2 Show Significant Efficacy in Delaying Tumor Growth.

2-氨基亚甲基-5-磺酰噻唑类赖氨酰氧化酶(LOX)和LOXL2抑制剂在延缓肿瘤生长方面显示出显著疗效

Smithen Deborah A, Leung Leo M H, Challinor Mairi, Lawrence Rae, Tang HaoRan, Niculescu-Duvaz Dan, Pearce Simon P, Mcleary Robert, Lopes Filipa, Aljarah Mohammed, Brown Michael, Johnson Louise, Thomson Graeme, Marais Richard, Springer Caroline

Paradox-breaking RAF inhibitors that also target SRC are effective in drug-resistant BRAF mutant melanoma

能够打破悖论且同时靶向SRC的RAF抑制剂对耐药性BRAF突变型黑色素瘤有效。

Girotti, Maria Romina; Lopes, Filipa; Preece, Natasha; Niculescu-Duvaz, Dan; Zambon, Alfonso; Davies, Lawrence; Whittaker, Steven; Saturno, Grazia; Viros, Amaya; Pedersen, Malin; Suijkerbuijk, Bart M J M; Menard, Delphine; McLeary, Robert; Johnson, Louise; Fish, Laura; Ejiama, Sarah; Sanchez-Laorden, Berta; Hohloch, Juliane; Carragher, Neil; Macleod, Kenneth; Ashton, Garry; Marusiak, Anna A; Fusi, Alberto; Brognard, John; Frame, Margaret; Lorigan, Paul; Marais, Richard; Springer, Caroline