日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Electrochemical deutero-(di)carboxylations for the preparation of deuterium-labeled medicinal building blocks

电化学氘代(二)羧化反应制备氘标记的药物结构单元

Mondal, Subhojit; Sahil; Brown, Alex; Meanwell, Michael W

Total Synthesis of Dragocins A-C through Electrochemical Cyclization

通过电化学环化法全合成Dragocins AC

Smith, Brendyn P; Truax, Nathanyal J; Pollatos, Alexandros S; Meanwell, Michael; Bedekar, Pranali; Garrido-Castro, Alberto F; Baran, Phil S

An enantioselective and modular platform for C4'-modified nucleoside analogue synthesis enabled by intramolecular trans-acetalizations

利用分子内转缩醛化反应实现的C4'修饰核苷类似物合成的对映选择性模块化平台

Nuligonda, Thirupathi; Kumar, Gautam; Wang, Jason W; Rajapaksha, Dinithi; Elayan, Ismael A; Demir, Ramiz; Meanwell, Neil J; Wang, Sherrie F; Mahal, Lara K; Brown, Alex; Meanwell, Michael W

N-Ammonium Ylide Mediators for Electrochemical C-H Oxidation

用于电化学CH氧化的N-铵叶立德介体

Saito, Masato; Kawamata, Yu; Meanwell, Michael; Navratil, Rafael; Chiodi, Debora; Carlson, Ethan; Hu, Pengfei; Chen, Longrui; Udyavara, Sagar; Kingston, Cian; Tanwar, Mayank; Tyagi, Sameer; McKillican, Bruce P; Gichinga, Moses G; Schmidt, Michael A; Eastgate, Martin D; Lamberto, Massimiliano; He, Chi; Tang, Tianhua; Malapit, Christian A; Sigman, Matthew S; Minteer, Shelley D; Neurock, Matthew; Baran, Phil S

Author Correction: Revealing the mechanism for covalent inhibition of glycoside hydrolases by carbasugars at an atomic level

作者更正:从原子层面揭示碳水化合物对糖苷水解酶的共价抑制机制

Ren, Weiwu; Pengelly, Robert; Farren-Dai, Marco; Abadi, Saeideh Shamsi Kazem; Oehler, Verena; Akintola, Oluwafemi; Draper, Jason; Meanwell, Michael; Chakladar, Saswati; Świderek, Katarzyna; Moliner, Vicent; Britton, Robert; Gloster, Tracey M; Bennet, Andrew J

Revealing the mechanism for covalent inhibition of glycoside hydrolases by carbasugars at an atomic level.

从原子水平揭示糖苷水解酶共价抑制的机制

Ren Weiwu, Pengelly Robert, Farren-Dai Marco, Shamsi Kazem Abadi Saeideh, Oehler Verena, Akintola Oluwafemi, Draper Jason, Meanwell Michael, Chakladar Saswati, Świderek Katarzyna, Moliner Vicent, Britton Robert, Gloster Tracey M, Bennet Andrew J

Direct heterobenzylic fluorination, difluorination and trifluoromethylthiolation with dibenzenesulfonamide derivatives

二苯磺酰胺衍生物的直接杂苄位氟化、二氟化和三氟甲基硫代化

Meanwell, Michael; Adluri, Bharani Shashank; Yuan, Zheliang; Newton, Josiah; Prevost, Philippe; Nodwell, Matthew B; Friesen, Chadron M; Schaffer, Paul; Martin, Rainer E; Britton, Robert