日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PEGylated Zein Micelles for Prostate Cancer Therapy: Influence of PEG Chain Length and Transferrin Targeting on Docetaxel Delivery

聚乙二醇化玉米醇溶蛋白胶束用于前列腺癌治疗:聚乙二醇链长度和转铁蛋白靶向对多西他赛递送的影响

Maeyouf, Khadeejah; Meewan, Jitkasem; Ali-Jerman, Hawraa; Albatsh, Musa; Somani, Sukrut; Laskar, Partha; Mullin, Margaret; Irving, Craig; MacKenzie, Graeme; Dufès, Christine

HBCVTr: an end-to-end transformer with a deep neural network hybrid model for anti-HBV and HCV activity predictor from SMILES

HBCVTr:一个端到端的Transformer模型,采用深度神经网络混合模型,用于预测基于SMILES的抗HBV和HCV活性。

Meewan, Ittipat; Panmanee, Jiraporn; Petchyam, Nopphon; Lertvilai, Pichaya

Transferrin-Bearing, Zein-Based Hybrid Lipid Nanoparticles for Drug and Gene Delivery to Prostate Cancer Cells

用于向前列腺癌细胞递送药物和基因的转铁蛋白负载玉米醇溶蛋白基混合脂质纳米颗粒

Maeyouf, Khadeejah; Sakpakdeejaroen, Intouch; Somani, Sukrut; Meewan, Jitkasem; Ali-Jerman, Hawraa; Laskar, Partha; Mullin, Margaret; MacKenzie, Graeme; Tate, Rothwelle J; Dufès, Christine

Allosteric Inhibitors of Zika Virus NS2B-NS3 Protease Targeting Protease in "Super-Open" Conformation

寨卡病毒NS2B-NS3蛋白酶的变构抑制剂靶向处于“超开放”构象的蛋白酶

Meewan, Ittipat; Shiryaev, Sergey A; Kattoula, Julius; Huang, Chun-Teng; Lin, Vivian; Chuang, Chiao-Han; Terskikh, Alexey V; Abagyan, Ruben

High-throughput phenotypic screen identifies a new family of potent anti-amoebic compounds

高通量表型筛选鉴定出一类新型强效抗阿米巴化合物

Sauvey, Conall; Meewan, Ittipat; Ehrenkaufer, Gretchen; Blevitt, Jonathan; Jackson, Paul; Abagyan, Ruben

Preparation of Zein-Based Nanoparticles: Nanoprecipitation versus Microfluidic-Assisted Manufacture, Effects of PEGylation on Nanoparticle Characteristics and Cellular Uptake by Melanoma Cells

玉米醇溶蛋白基纳米粒子的制备:纳米沉淀与微流体辅助制造、聚乙二醇化对纳米粒子特性的影响以及黑色素瘤细胞的细胞摄取

Jitkasem Meewan, Sukrut Somani, Jamal Almowalad, Partha Laskar, Margaret Mullin, Graeme MacKenzie, Swapnil Khadke, Yvonne Perrie, Christine Dufès

Lactoferrin- and Dendrimer-Bearing Gold Nanocages for Stimulus-Free DNA Delivery to Prostate Cancer Cells

载有乳铁蛋白和树枝状聚合物的金纳米笼用于无刺激 DNA 递送至前列腺癌细胞

Jamal Almowalad, Partha Laskar, Sukrut Somani, Jitkasem Meewan, Rothwelle J Tate, Christine Dufès

Limited Impact of the Protein Corona on the Cellular Uptake of PEGylated Zein Micelles by Melanoma Cancer Cells

蛋白冠对黑色素瘤癌细胞摄取聚乙二醇化玉米醇溶蛋白胶束的影响有限

Jitkasem Meewan, Sukrut Somani, Partha Laskar, Craig Irving, Margaret Mullin, Stuart Woods, Craig W Roberts, Abdullah R Alzahrani, Valerie A Ferro, Suzanne McGill, Stefan Weidt, Richard Burchmore, Christine Dufès

Discovery of Triple Inhibitors of Both SARS-CoV-2 Proteases and Human Cathepsin L

发现 SARS-CoV-2 蛋白酶和人类组织蛋白酶 L 的三重抑制剂

Ittipat Meewan, Jacob Kattoula, Julius Y Kattoula, Danielle Skinner, Pavla Fajtová, Miriam A Giardini, Brendon Woodworth, James H McKerrow, Jair Lage de Siqueira-Neto, Anthony J O'Donoghue, Ruben Abagyan

Phenotypic, chemical and functional characterization of cyclic nucleotide phosphodiesterase 4 (PDE4) as a potential anthelmintic drug target.

环核苷酸磷酸二酯酶 4 (PDE4) 作为潜在驱虫药物靶点的表型、化学和功能表征

Long Thavy, Rojo-Arreola Liliana, Shi Da, El-Sakkary Nelly, Jarnagin Kurt, Rock Fernando, Meewan Maliwan, Rascón Alberto A Jr, Lin Lin, Cunningham Katherine A, Lemieux George A, Podust Larissa, Abagyan Ruben, Ashrafi Kaveh, McKerrow James H, Caffrey Conor R