日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanism-Based Inactivation of Cytochrome P450 3A4 and 3A5 by the Fibroblast Growth Factor Receptor Inhibitor Erdafitinib

成纤维细胞生长因子受体抑制剂厄达替尼基于机制地灭活细胞色素 P450 3A4 和 3A5

Lloyd Wei Tat Tang, Jian Wei Teng, Siew Kwan Koh, Lei Zhou, Mei Lin Go, Eric Chun Yong Chan

Extreme Drug Tolerance of Mycobacterium abscessus "Persisters"

脓肿分枝杆菌“持久菌”的极强耐药性

Yee-Kuen Yam, Nadine Alvarez, Mei-Lin Go, Thomas Dick

Gut Microbiota Metabolite Indole Propionic Acid Targets Tryptophan Biosynthesis in Mycobacterium tuberculosis

肠道微生物代谢物吲哚丙酸靶向结核分枝杆菌中的色氨酸生物合成

Dereje Abate Negatu, Yoshiyuki Yamada, Yu Xi, Mei Lin Go, Matthew Zimmerman, Uday Ganapathy, Véronique Dartois, Martin Gengenbacher, Thomas Dick

Indolyl Azaspiroketal Mannich Bases Are Potent Antimycobacterial Agents with Selective Membrane Permeabilizing Effects and in Vivo Activity

吲哚基氮杂螺酮 Mannich 碱是具有选择性膜通透作用和体内活性的强效抗分枝杆菌剂

Samuel Agyei Nyantakyi, Ming Li, Pooja Gopal, Matthew Zimmerman, Véronique Dartois, Martin Gengenbacher, Thomas Dick, Mei-Lin Go

A New Generation of Arachidonic Acid Analogues as Potential Neurological Agent Targeting Cytosolic Phospholipase A2

新一代花生四烯酸类似物作为靶向胞浆磷脂酶 A2 的潜在神经药物

Cheng Yang Ng, Srinivasaraghavan Kannan, Yong Jun Chen, Francis Chee Kuan Tan, Wee Yong Ong, Mei Lin Go, Chandra S Verma, Chian-Ming Low, Yulin Lam

Dioxonaphthoimidazoliums AB1 and YM155 disrupt phosphorylation of p50 in the NF-κB pathway

二氧萘并咪唑鎓 AB1 和 YM155 破坏 NF-κB 通路中 p50 的磷酸化

Si Han Sherman Ho, Azhar Ali, Tan Min Chin, Mei Lin Go

Functionalized tetrahydro-1H-pyrido[4,3-b]indoles: a novel chemotype with Sirtuin 2 inhibitory activity

功能化四氢-1H-吡啶并[4,3-b]吲哚:具有 Sirtuin 2 抑制活性的新型化学类型

Tianming Yang, Xiao Chen, Hai-xiao Jin, Gautam Sethi, Mei-Lin Go

Synthesis and evaluation of bisbenzylidenedioxotetrahydrothiopranones as activators of endoplasmic reticulum (ER) stress signaling pathways and apoptotic cell death in acute promyelocytic leukemic cells

双苄基二氧代四氢噻吩酮的合成及作为内质网 (ER) 应激信号通路激活剂和急性早幼粒白血病细胞凋亡的细胞死亡的评价

Kheng-Lin Tan, Azhar Ali, Yuhong Du, Haian Fu, Hai-Xiao Jin, Tan-Min Chin, Matiullah Khan, Mei-Lin Go

An improved isoprenylcysteine carboxylmethyltransferase inhibitor induces cancer cell death and attenuates tumor growth in vivo

改进的异戊二烯半胱氨酸羧甲基转移酶抑制剂可诱导癌细胞死亡并减弱体内肿瘤生长

Hiu Yeung Lau, Pondy M Ramanujulu, Dianyan Guo, Tianming Yang, Melissa Wirawan, Patrick J Casey, Mei-Lin Go, Mei Wang

Structural characterization of myotoxic ecarpholin S from Echis carinatus venom

锯鳞蝰毒中肌毒性 Ecarpholin S 的结构表征

Xingding Zhou, Tien-Chye Tan, S Valiyaveettil, Mei Lin Go, R Manjunatha Kini, Adrian Velazquez-Campoy, J Sivaraman