Discovery of Potent PDE4 Inhibitors with 3(2H)-Pyridazinone Scaffold: Synthesis, In Silico Studies and In Vitro/Vivo Evaluation
发现具有3(2H)-哒嗪酮骨架的高效PDE4抑制剂:合成、计算机模拟研究和体外/体内评价
期刊:Molecules
影响因子:4.6
doi:10.3390/molecules31040699
Vergelli, Claudia; Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Gracia, Jordi; Buil, Maria Antonia; Garrido, Yolanda; Pagès, Lluis; Taltavull, Joan; Gavaldà, Amadeu; Calama, Elena; Giovannoni, Maria Paola