日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of Potent PDE4 Inhibitors with 3(2H)-Pyridazinone Scaffold: Synthesis, In Silico Studies and In Vitro/Vivo Evaluation

发现具有3(2H)-哒嗪酮骨架的高效PDE4抑制剂:合成、计算机模拟研究和体外/体内评价

Vergelli, Claudia; Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Gracia, Jordi; Buil, Maria Antonia; Garrido, Yolanda; Pagès, Lluis; Taltavull, Joan; Gavaldà, Amadeu; Calama, Elena; Giovannoni, Maria Paola

Synthesis of 3-Carboxy-6-sulfamoylquinolones and Mefloquine-Based Compounds as Panx1 Blockers: Molecular Docking, Electrophysiological and Cell Culture Studies

3-羧基-6-氨磺酰喹诺酮类化合物和甲氟喹类化合物作为Panx1阻滞剂的合成:分子对接、电生理和细胞培养研究

Crocetti, Letizia; Giovannoni, Maria Paola; Pavlov, Tengis S; Ivanov, Veniamin; Melani, Fabrizio; Guerrini, Gabriella

Anti-Inflammatory Activity of Pyrazolo[1,5-a]quinazolines

吡唑并[1,5-a]喹唑啉的抗炎活性

Crocetti, Letizia; Khlebnikov, Andrei I; Guerrini, Gabriella; Schepetkin, Igor A; Melani, Fabrizio; Giovannoni, Maria Paola; Quinn, Mark T

Design, Synthesis and Pharmacological Evaluation of New Quinoline-Based Panx-1 Channel Blockers

新型喹啉类Panx-1通道阻滞剂的设计、合成及药理学评价

Crocetti, Letizia; Giovannoni, Maria Paola; Guerrini, Gabriella; Lamanna, Silvia; Melani, Fabrizio; Bartolucci, Gianluca; Pallecchi, Marco; Paoli, Paola; Lippi, Martina; Wang, Junjie; Dahl, Gerhard

4,5-Dihydro-5-Oxo-Pyrazolo[1,5-a]Thieno[2,3-c]Pyrimidine: A Novel Scaffold Containing Thiophene Ring. Chemical Reactivity and In Silico Studies to Predict the Profile to GABA(A) Receptor Subtype

4,5-二氢-5-氧代-吡唑并[1,5-a]噻吩并[2,3-c]嘧啶:一种新型含噻吩环的骨架。化学反应性和计算机模拟研究预测其对GABA(A)受体亚型的亲和力。

Crocetti, Letizia; Guerrini, Gabriella; Melani, Fabrizio; Vergelli, Claudia; Giovannoni, Maria Paola

New Panx-1 Blockers: Synthesis, Biological Evaluation and Molecular Dynamic Studies.

新型 Panx-1 阻滞剂:合成、生物学评价和分子动力学研究

Crocetti Letizia, Guerrini Gabriella, Giovannoni Maria Paola, Melani Fabrizio, Lamanna Silvia, Di Cesare Mannelli Lorenzo, Lucarini Elena, Ghelardini Carla, Wang Junjie, Dahl Gerhard

4-Heteroaryl Substituted Amino-3,5-Dicyanopyridines as New Adenosine Receptor Ligands: Novel Insights on Structure-Activity Relationships and Perspectives

4-杂芳基取代的氨基-3,5-二氰基吡啶作为新型腺苷受体配体:结构-活性关系的新见解和展望

Catarzi, Daniela; Varano, Flavia; Vigiani, Erica; Calenda, Sara; Melani, Fabrizio; Varani, Katia; Vincenzi, Fabrizio; Pasquini, Silvia; Mennini, Natascia; Nerli, Giulia; Dal Ben, Diego; Volpini, Rosaria; Colotta, Vittoria

Combined Use of Cyclodextrins and Amino Acids for the Development of Cefixime Oral Solutions for Pediatric Use

环糊精与氨基酸联合用于开发儿童用头孢克肟口服溶液

Cirri, Marzia; Mennini, Natascia; Nerli, Giulia; Rubia, Jessica; Casalone, Enrico; Melani, Fabrizio; Maestrelli, Francesca; Mura, Paola