日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Biological Activity of Novel Ornithine Decarboxylase (ODC) Inhibitors

新型鸟氨酸脱羧酶(ODC)抑制剂的设计、合成及生物活性

Schultz, Chad R; Aleiwi, Bilal; Zhou, X Edward; Suino-Powell, Kelly; Melcher, Karsten; Almeida, Nuno M S; Wilson, Angela K; Ellsworth, Edmund L; Bachmann, André S

Assembly of JAZ-JAZ and JAZ-NINJA complexes in jasmonate signaling

茉莉酸信号传导中 JAZ-JAZ 和 JAZ-NINJA 复合物的组装

Zhou, X Edward; Zhang, Yaguang; Yao, Jian; Zheng, Jie; Zhou, Yuxin; He, Qing; Moreno, Javier; Lam, Vinh Q; Cao, Xiaoman; Sugimoto, Koichi; Vanegas-Cano, Leidy; Kariapper, Leena; Suino-Powell, Kelly; Zhu, Yuanye; Novick, Scott; Griffin, Patrick R; Zhang, Feng; Howe, Gregg A; Melcher, Karsten

Structure insights into selective coupling of G protein subtypes by a class B G protein-coupled receptor.

通过BG类蛋白偶联受体对G蛋白亚型进行选择性偶联的结构解析

Zhao Li-Hua, Lin Jingyu, Ji Su-Yu, Zhou X Edward, Mao Chunyou, Shen Dan-Dan, He Xinheng, Xiao Peng, Sun Jinpeng, Melcher Karsten, Zhang Yan, Yu Xiao, Xu H Eric

Structure of an AMPK complex in an inactive, ATP-bound state

处于非活性、ATP结合状态的AMPK复合物的结构

Yan, Yan; Mukherjee, Somnath; Harikumar, Kaleeckal G; Strutzenberg, Timothy S; Zhou, X Edward; Suino-Powell, Kelly; Xu, Ting-Hai; Sheldon, Ryan D; Lamp, Jared; Brunzelle, Joseph S; Radziwon, Katarzyna; Ellis, Abigail; Novick, Scott J; Vega, Irving E; Jones, Russell G; Miller, Laurence J; Xu, H Eric; Griffin, Patrick R; Kossiakoff, Anthony A; Melcher, Karsten

Long-chain fatty acyl-CoA esters regulate metabolism via allosteric control of AMPK β1 isoforms.

长链脂肪酰辅酶A酯通过变构控制AMPK β1同工酶来调节代谢

Pinkosky Stephen L, Scott John W, Desjardins Eric M, Smith Brennan K, Day Emily A, Ford Rebecca J, Langendorf Christopher G, Ling Naomi X Y, Nero Tracy L, Loh Kim, Galic Sandra, Hoque Ashfaqul, Smiles William J, Ngoei Kevin R W, Parker Michael W, Yan Yan, Melcher Karsten, Kemp Bruce E, Oakhill Jonathan S, Steinberg Gregory R

Identification and structural insight of an effective PPARγ modulator with improved therapeutic index for anti-diabetic drug discovery

鉴定并解析一种具有更高治疗指数的有效PPARγ调节剂的结构,用于抗糖尿病药物研发

Jiang, Haowen; Zhou, X Edward; Shi, Jingjing; Zhou, Zhi; Zhao, Guanguan; Zhang, Xinwen; Sun, Yili; Suino-Powell, Kelly; Ma, Lei; Gao, Hui; Yu, Xiyong; Li, Jia; Li, Jingya; Melcher, Karsten; Xu, H Eric; Yi, Wei

Molecular mechanisms of fentanyl mediated β-arrestin biased signaling

芬太尼介导的β-arrestin偏向性信号的分子机制

de Waal, Parker W; Shi, Jingjing; You, Erli; Wang, Xiaoxi; Melcher, Karsten; Jiang, Yi; Xu, H Eric; Dickson, Bradley M

Structure and dynamics of the active human parathyroid hormone receptor-1

活性人甲状旁腺激素受体-1的结构和动力学

Zhao, Li-Hua; Ma, Shanshan; Sutkeviciute, Ieva; Shen, Dan-Dan; Zhou, X Edward; de Waal, Parker W; Li, Chen-Yao; Kang, Yanyong; Clark, Lisa J; Jean-Alphonse, Frederic G; White, Alex D; Yang, Dehua; Dai, Antao; Cai, Xiaoqing; Chen, Jian; Li, Cong; Jiang, Yi; Watanabe, Tomoyuki; Gardella, Thomas J; Melcher, Karsten; Wang, Ming-Wei; Vilardaga, Jean-Pierre; Xu, H Eric; Zhang, Yan

Structural biology of G protein-coupled receptor signaling complexes

G蛋白偶联受体信号复合物的结构生物学

Edward Zhou, X; Melcher, Karsten; Eric Xu, H

Crystal structure of the human 5-HT(1B) serotonin receptor bound to an inverse agonist

人5-HT(1B)血清素受体与反向激动剂结合的晶体结构

Yin, Wanchao; Zhou, X Edward; Yang, Dehua; de Waal, Parker W; Wang, Meitian; Dai, Antao; Cai, Xiaoqing; Huang, Chia-Ying; Liu, Ping; Wang, Xiaoxi; Yin, Yanting; Liu, Bo; Zhou, Yu; Wang, Jiang; Liu, Hong; Caffrey, Martin; Melcher, Karsten; Xu, Yechun; Wang, Ming-Wei; Xu, H Eric; Jiang, Yi