Tonabersat enhances temozolomide-mediated cytotoxicity in glioblastoma by disrupting intercellular connectivity through connexin 43 inhibition.
Tonabersat 通过抑制连接蛋白 43 来破坏细胞间连接,从而增强替莫唑胺对胶质母细胞瘤的细胞毒性
期刊:Molecular Oncology
影响因子:4.5
doi:10.1002/1878-0261.13786
Schmidt Elena N C, Evert Bernd O, Pregler Barbara E F, Melhem Ahmad, Hsieh Meng-Chun, Raspe Markus, Strobel Hannah, Roos Julian, Pietsch Torsten, Schuss Patrick, Fischer-Posovszky Pamela, Westhoff Mike-Andrew, Hölzel Michael, Herrlinger Ulrich, Vatter Hartmut, Waha Andreas, Schneider Matthias, Potthoff Anna-Laura