Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation
设计、合成和生物学评价喹啉类化合物SGI-1027的4-氨基-N-(4-氨基苯基)苯甲酰胺类似物作为DNA甲基化抑制剂
期刊:ChemMedChem
影响因子:3.4
doi:10.1002/cmdc.201300420
Rilova, Elodie; Erdmann, Alexandre; Gros, Christina; Masson, Véronique; Aussagues, Yannick; Poughon-Cassabois, Valérie; Rajavelu, Arumugam; Jeltsch, Albert; Menon, Yoann; Novosad, Natacha; Gregoire, Jean-Marc; Vispé, Stéphane; Schambel, Philippe; Ausseil, Fréderic; Sautel, François; Arimondo, Paola B; Cantagrel, Frédéric