日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, synthesis and biological evaluation of 4-amino-N- (4-aminophenyl)benzamide analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation

设计、合成和生物学评价喹啉类化合物SGI-1027的4-氨基-N-(4-氨基苯基)苯甲酰胺类似物作为DNA甲基化抑制剂

Rilova, Elodie; Erdmann, Alexandre; Gros, Christina; Masson, Véronique; Aussagues, Yannick; Poughon-Cassabois, Valérie; Rajavelu, Arumugam; Jeltsch, Albert; Menon, Yoann; Novosad, Natacha; Gregoire, Jean-Marc; Vispé, Stéphane; Schambel, Philippe; Ausseil, Fréderic; Sautel, François; Arimondo, Paola B; Cantagrel, Frédéric

Development of a universal radioactive DNA methyltransferase inhibition test for high-throughput screening and mechanistic studies.

开发一种通用的放射性DNA甲基转移酶抑制试验,用于高通量筛选和机制研究

Gros Christina, Chauvigné Laura, Poulet Anaïs, Menon Yoann, Ausseil Frédéric, Dufau Isabelle, Arimondo Paola B