文献库，生知库 | 链接生命科学的每一步

日期影响因子

Hydrogen-bonded His93 as a sensitive probe for identifying inhibitors of the endocannabinoid transport protein FABP7.

氢键结合的 His93 可作为识别内源性大麻素转运蛋白 FABP7 抑制剂的敏感探针

期刊:Chemical Biology & Drug Design

影响因子:3.3

doi:10.1111/cbdd.12440

Tyukhtenko Sergiy, Chan Karrie, Jiang Rubin, Zhou Han, Mercier Richard W, Yang De-Ping, Makriyannis Alexandros, Guo Jason J

发表日期：2015

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Assay and inhibition of diacylglycerol lipase activity

二酰甘油脂肪酶活性的测定和抑制

期刊:Bioorganic & Medicinal Chemistry Letters

影响因子:2.2

doi:10.1016/j.bmcl.2012.05.101

Johnston, Meghan; Bhatt, Shachi R; Sikka, Surina; Mercier, Richard W; West, Jay M; Makriyannis, Alexandros; Gatley, S John; Duclos, Richard I Jr

发表日期：2012

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Mass spectrometry-based proteomics of human cannabinoid receptor 2: covalent cysteine 6.47(257)-ligand interaction affording megagonist receptor activation.

基于质谱的人类大麻素受体 2 蛋白质组学：半胱氨酸 6.47(257)-配体共价相互作用可激活巨激动剂受体

期刊:Journal of Proteome Research

影响因子:3.6

doi:10.1021/pr2005583

Szymanski Dennis W, Papanastasiou Malvina, Melchior Katja, Zvonok Nikolai, Mercier Richard W, Janero David R, Thakur Ganesh A, Cha Sangwon, Wu Billy, Karger Barry, Makriyannis Alexandros

免疫/内分泌

发表日期：2011

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hCB2 ligand-interaction landscape: cysteine residues critical to biarylpyrazole antagonist binding motif and receptor modulation

hCB2配体相互作用图谱：对联芳基吡唑拮抗剂结合基序和受体调控至关重要的半胱氨酸残基

doi:10.1016/j.chembiol.2010.08.010

Mercier, Richard W; Pei, Ying; Pandarinathan, Lakshmipathi; Janero, David R; Zhang, Jing; Makriyannis, Alexandros

发表日期：2010

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Ligand-binding architecture of human CB2 cannabinoid receptor: evidence for receptor subtype-specific binding motif and modeling GPCR activation

人CB2大麻素受体的配体结合结构：受体亚型特异性结合基序的证据及GPCR激活建模

doi:10.1016/j.chembiol.2008.10.011

Pei, Ying; Mercier, Richard W; Anday, Jenine K; Thakur, Ganesh A; Zvonok, Alexander M; Hurst, Dow; Reggio, Patricia H; Janero, David R; Makriyannis, Alexandros

GPCR/Calcium/cAMP

发表日期：2008

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Interaction of a fragment of the cannabinoid CB1 receptor C-terminus with arrestin-2

大麻素 CB1 受体 C 端片段与阻遏蛋白-2 的相互作用

doi:10.1016/j.febslet.2007.09.030

Bakshi, Kunal; Mercier, Richard W; Pavlopoulos, Spiro

发表日期：2007

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