Tranylcypromine-Based LSD1 Inhibitors: Structure-Activity Relationships, Antiproliferative Effects in Leukemia, and Gene Target Modulation
基于反苯环丙胺的 LSD1 抑制剂:结构-活性关系、白血病中的抗增殖作用和基因靶标调节
期刊:ChemMedChem
影响因子:3.6
doi:10.1002/cmdc.201900730
Rossella Fioravanti, Annalisa Romanelli, Nicola Mautone, Elisabetta Di Bello, Annarita Rovere, Davide Corinti, Clemens Zwergel, Sergio Valente, Dante Rotili, Oronza A Botrugno, Paola Dessanti, Stefania Vultaggio, Paola Vianello, Anna Cappa, Claudia Binda, Andrea Mattevi, Saverio Minucci, Ciro Mercur