日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

First-in-Human Clinical Trial of a Small-Molecule EBNA1 Inhibitor, VK-2019, in Patients with Epstein-Barr-Positive Nasopharyngeal Cancer, with Pharmacokinetic and Pharmacodynamic Studies.

首次对 Epstein-Barr 阳性鼻咽癌患者进行小分子 EBNA1 抑制剂 VK-2019 的人体临床试验,并进行药代动力学和药效学研究

Colevas A Dimitrios, Talebi Zahra, Winters Elizabeth, Even Caroline, Lee Victor Ho-Fun, Gillison Maura L, Khan Saad A, Lu Rong, Pinsky Benjamin A, Soldan Samantha S, Vladmirova Olga, Lieberman Paul M, Messick Troy E

Metabolomic Analysis and Antiviral Screening of a Marine Algae Library Yield Jobosic Acid (2,5-Dimethyltetradecanoic Acid) as a Selective Inhibitor of SARS-CoV-2.

对海洋藻类库进行代谢组学分析和抗病毒筛选,发现乔博西酸(2,5-二甲基十四烷酸)是SARS-CoV-2的选择性抑制剂

Matos-Hernández Marie L, Samples Robert, Dyer Grayce, Casimir Montán Victoria M, Morales-Colón Chris A, Salvino Joseph M, Montaner Luis J, Cassel Joel A, Messick Troy E, Tietjen Ian, Caro-Diaz Eduardo J E

Therapeutic approaches to Epstein-Barr virus cancers

治疗EB病毒相关癌症的方法

Soldan, Samantha S; Messick, Troy E; Lieberman, Paul M

Cryo-EM Structure and Functional Studies of EBNA1 Binding to the Family of Repeats and Dyad Symmetry Elements of Epstein-Barr Virus oriP.

EBNA1 与 Epstein-Barr 病毒 oriP 的重复序列和二元对称元件家族结合的冷冻电镜结构和功能研究

Mei Yang, Messick Troy E, Dheekollu Jayaraju, Kim Hee Jong, Molugu Sudheer, Muñoz Leonardo Josué Castro, Moiskeenkova-Bell Vera, Murakami Kenji, Lieberman Paul M

EBNA1 inhibitors have potent and selective antitumor activity in xenograft models of Epstein-Barr virus-associated gastric cancer

EBNA1抑制剂在Epstein-Barr病毒相关胃癌异种移植模型中具有强效且选择性的抗肿瘤活性。

Soldan, Samantha S; Anderson, Emma M; Frase, Drew M; Zhang, Yue; Caruso, Lisa B; Wang, Yin; Deakyne, Julianna S; Gewurz, Benjamin E; Tempera, Italo; Lieberman, Paul M; Messick, Troy E

Correction: Carcinoma-risk variant of EBNA1 deregulates Epstein-Barr Virus episomal latency

更正:EBNA1 的致癌风险变异体可解除 Epstein-Barr 病毒游离型潜伏的调控。

Dheekollu, Jayaraju; Malecka, Kimberly; Wiedmer, Andreas; Delecluse, Henri-Jacques; Chiang, Alan K S; Altieri, Dario C; Messick, Troy E; Lieberman, Paul M

Biallelic deleterious BRCA1 mutations in a woman with early-onset ovarian cancer

一名患有早发性卵巢癌的女性携带双等位基因有害的BRCA1突变

Domchek, Susan M; Tang, Jiangbo; Stopfer, Jill; Lilli, Dana R; Hamel, Nancy; Tischkowitz, Marc; Monteiro, Alvaro N A; Messick, Troy E; Powers, Jacquelyn; Yonker, Alexandria; Couch, Fergus J; Goldgar, David E; Davidson, H Rosemarie; Nathanson, Katherine L; Foulkes, William D; Greenberg, Roger A

Crystal structure and functional interpretation of the erythrocyte spectrin tetramerization domain complex

红细胞血影蛋白四聚体化结构域复合物的晶体结构及功能解析

Ipsaro, Jonathan J; Harper, Sandra L; Messick, Troy E; Marmorstein, Ronen; Mondragón, Alfonso; Speicher, David W

The ubiquitin landscape at DNA double-strand breaks

DNA双链断裂处的泛素分布

Messick, Troy E; Greenberg, Roger A