日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Synthetic chemistry enabling the discovery and development of a series of pyrazoles as HPK1 inhibitors

合成化学促进了一系列吡唑类化合物作为HPK1抑制剂的发现和开发

Metrano, Anthony J; Morrill, Lucas A; Bommakanti, Gayathri; Casella, Robert; Cook, Steve; Escobar, Randolph A; Giblin, Kathryn A; Gosselin, Eric; Grebe, Tyler; Hariparsad, Niresh; Howells, Rachel; Lamont, Gillian M; Mele, Deanna A; Pflug, Alexander; Proia, Theresa A; Rezaei, Hadi; Richter, Magdalena; Richards, Ryan; San Martin, Maryann; Schimpl, Marianne; Schuller, Alwin G; Sha, Li; Sheppeck, James E 2nd; Song, Kun; Tang, Haoran; Wagner, David J; Wang, Jianyan; Wu, Allan; Wu, Dedong; Wu, Ye; Xu, Kevin; Ye, Minwei; Shields, Jason D; Grimster, Neil P

Isolating Conformers to Assess Dynamics of Peptidic Catalysts Using Computationally Designed Macrocyclic Peptides

利用计算机设计的环状肽分离构象异构体以评估肽催化剂的动力学

Stone, Elizabeth A; Hosseinzadeh, Parisa; Craven, Timothy W; Robertson, Michael J; Han, Yaodong; Hsieh, Sheng-Ying; Metrano, Anthony J; Baker, David; Miller, Scott J

Asymmetric Catalysis Mediated by Synthetic Peptides, Version 2.0: Expansion of Scope and Mechanisms

合成肽介导的不对称催化,2.0版:范围和机制的扩展

Metrano, Anthony J; Chinn, Alex J; Shugrue, Christopher R; Stone, Elizabeth A; Kim, Byoungmoo; Miller, Scott J

Peptide-Based Catalysts Reach the Outer Sphere through Remote Desymmetrization and Atroposelectivity

基于肽的催化剂通过远程去对称化和阻转选择性到达外层

Metrano, Anthony J; Miller, Scott J

Troponoid Atropisomerism: Studies on the Configurational Stability of Tropone-Amide Chiral Axes

环庚三烯酮类化合物的阻转异构现象:环庚三烯酮-酰胺手性轴构型稳定性的研究

Hirsch, Danielle R; Metrano, Anthony J; Stone, Elizabeth A; Storch, Golo; Miller, Scott J; Murelli, Ryan P

Parameterization and Analysis of Peptide-Based Catalysts for the Atroposelective Bromination of 3-Arylquinazolin-4(3H)-ones

肽基催化剂对3-芳基喹唑啉-4(3H)-酮的阻转选择性溴化反应的参数化和分析

Crawford, Jennifer M; Stone, Elizabeth A; Metrano, Anthony J; Miller, Scott J; Sigman, Matthew S

Molecular Dynamics Simulations of a Conformationally Mobile Peptide-Based Catalyst for Atroposelective Bromination

利用分子动力学模拟研究构象可移动的肽基催化剂在对映选择性溴化反应中的应用

Yan, Xin Cindy; Metrano, Anthony J; Robertson, Michael J; Abascal, Nadia C; Tirado-Rives, Julian; Miller, Scott J; Jorgensen, William L

Diversity of Secondary Structure in Catalytic Peptides with β-Turn-Biased Sequences

具有β-转角偏向序列的催化肽二级结构的多样性

Metrano, Anthony J; Abascal, Nadia C; Mercado, Brandon Q; Paulson, Eric K; Hurtley, Anna E; Miller, Scott J

Spontaneous transfer of chirality in an atropisomerically enriched two-axis system

在富含阻转异构体的双轴体系中手性的自发转移

Barrett, Kimberly T; Metrano, Anthony J; Rablen, Paul R; Miller, Scott J