日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of SD-965 as a Potent, Selective, and Efficacious STAT3 PROTAC Degrader

发现 SD-965 是一种高效、选择性强且有效的 STAT3 PROTAC 降解剂

Wu, Dimin; Zhou, Haibin; Bai, Longchuan; Acharyya, Ranjan Kumar; Metwally, Hoda; McEachern, Donna; Wang, Mi; Tošović, Jelena; Rej, Rohan Kalyan; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng

MD-4251: A First-in-Class Oral MDM2 Degrader Inducing Complete Tumor Regression with Single-Dose Administration

MD-4251:一种首创的口服MDM2降解剂,单次给药即可诱导肿瘤完全消退

Acharyya, Ranjan Kumar; Huang, Liyue; Aguilar, Angelo; Hu, Biao; Bai, Longchuan; Metwally, Hoda; McEachern, Donna; Jiang, Wei; Wang, Yu; Li, Qiuxia; Wen, Bo; Sun, Duxin; Wang, Shaomeng

Discovery of ERD-1233 as a Potent and Orally Efficacious Estrogen Receptor PROTAC Degrader for the Treatment of ER+ Human Breast Cancer

发现 ERD-1233 是一种强效且口服有效的雌激素受体 PROTAC 降解剂,可用于治疗 ER+ 人类乳腺癌

Acharyya, Ranjan Kumar; Rej, Rohan Kalyan; Hu, Biao; Chen, Zhixiang; Wu, Dimin; Lu, Jianfeng; Metwally, Hoda; McEachern, Donna; Wang, Yu; Jiang, Wei; Bai, Longchuan; Tošović, Jelena; Gersch, Christina L; Xu, Guozhang; Zhang, Weihong; Wu, WenXue; Priestley, E Scott; Sui, Zhihua; Sarkari, Farzad; Wen, Bo; Sun, Duxin; Rae, James M; Wang, Shaomeng

Discovery of ERD-12310A as an Exceptionally Potent and Orally Efficacious PROTAC Degrader of Estrogen Receptor α (ERα).

发现 ERD-12310A 是一种效力极强且口服有效的雌激素受体 α (ERα) PROTAC 降解剂。

Rej Rohan Kalyan, Hu Biao, Chen Zhixiang, Acharyya Ranjan Kumar, Wu Dimin, Metwally Hoda, McEachern Donna, Wang Yu, Jiang Wei, Bai Longchuan, Nishimura Leticia S, Gersch Christina L, Wang Meilin, Wen Bo, Sun Duxin, Carlson Kathryn, Katzenellenbogen John A, Xu Guozhang, Zhang Weihong, Wu Wenxue, Priestley E Scott, Sui Zhihua, Rae James M, Wang Shaomeng

Discovery of ARD-2585 as an Exceptionally Potent and Orally Active PROTAC Degrader of Androgen Receptor for the Treatment of Advanced Prostate Cancer.

发现 ARD-2585 是一种效力极强且口服有效的 PROTAC 雄激素受体降解剂,可用于治疗晚期前列腺癌

Xiang Weiguo, Zhao Lijie, Han Xin, Qin Chong, Miao Bukeyan, McEachern Donna, Wang Yu, Metwally Hoda, Kirchhoff Paul D, Wang Lu, Matvekas Aleksas, He Miao, Wen Bo, Sun Duxin, Wang Shaomeng