日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Anti-pyroglutamate-3 Aβ immunotherapy engages microglia and inhibits amyloid accumulation in transgenic mouse models of Aβ amyloidosis.

抗焦谷氨酸-3 Aβ 免疫疗法可激活小胶质细胞,并抑制 Aβ 淀粉样变性转基因小鼠模型中的淀粉样蛋白积累

Liao Fan, Calvo-Rodriguez Maria, Chhaya Meha, Sefrin Julian P, Charych Erik I, Mezler Mario, Clausznitzer Diana, McGlame Emily J, Zhao Karen, Rodgers Allison, Cao Yang, Secker Philipp F, Fernandez Garcia-Agudo Laura, Huang Lili, Klein Corinna, Dellovade Tammy, Karran Eric

Cortical organoid-derived models of the melanoma brain metastatic niche enable prioritization of cancer-targeting drugs.

利用皮质类器官衍生的黑色素瘤脑转移微环境模型,可以对癌症靶向药物进行优先排序。

Krieg Kim, Materna-Reichelt Silvia, Naber Tobias, Rachad Fatima-Zahra, Kauven Pia, Weller Arjen, Haferkamp Undine, Wittich Annika, Zaliani Andrea, Woo Marcel S, Walkenhorst Mark, Siegmund Malte, Harberts Jann, Zierold Robert, Blick Robert, Conze Christian, Muschong Patricia, Miltner Dominik, Friese Manuel A, Mezler Mario, Siegmund Heiko, Evert Katja, Krasemann Susanne, Gužvić Nataša Stojanović, Klein Christoph A, Werner-Klein Melanie, Wegener Joachim, Pless Ole

Conquering the beyond Rule of Five Space with an Optimized High-Throughput Caco-2 Assay to Close Gaps in Absorption Prediction

利用优化的高通量Caco-2检测方法攻克“五规则”之外的领域,以弥补吸收预测方面的差距

Muschong, Patricia; Awwad, Khader; Price, Edward; Mezler, Mario; Weinheimer, Manuel

Challenges in Permeability Assessment for Oral Drug Product Development

口服药物产品开发中渗透性评估的挑战

Koziolek, Mirko; Augustijns, Patrick; Berger, Constantin; Cristofoletti, Rodrigo; Dahlgren, David; Keemink, Janneke; Matsson, Pär; McCartney, Fiona; Metzger, Marco; Mezler, Mario; Niessen, Janis; Polli, James E; Vertzoni, Maria; Weitschies, Werner; Dressman, Jennifer

Novel Developments to Enable Treatment of CNS Diseases with Targeted Drug Delivery

利用靶向药物递送治疗中枢神经系统疾病的新进展

Meyer, Axel H; Feldsien, Thomas M; Mezler, Mario; Untucht, Christopher; Venugopalan, Ramakrishna; Lefebvre, Didier R

Mucin-Protected Caco-2 Assay to Study Drug Permeation in the Presence of Complex Biorelevant Media

利用粘蛋白保护的Caco-2细胞测定法研究复杂生物相关介质中药物的渗透性

Ye, Dong; López Mármol, Álvaro; Lenz, Verena; Muschong, Patricia; Wilhelm-Alkubaisi, Anita; Weinheimer, Manuel; Koziolek, Mirko; Sauer, Kerstin A; Laplanche, Loic; Mezler, Mario