Discovery of a potent and highly selective PDK1 inhibitor via fragment-based drug discovery
通过基于片段的药物发现发现有效且高选择性的 PDK1 抑制剂
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.5
doi:10.1016/j.bmcl.2011.03.032
Daniel A Erlanson, Joseph W Arndt, Mark T Cancilla, Kathy Cao, Robert A Elling, Nicki English, Jessica Friedman, Stig K Hansen, Cathy Hession, Ingrid Joseph, Gnanasambandam Kumaravel, Wen-Cherng Lee, Ken E Lind, Robert S McDowell, Konrad Miatkowski, Christine Nguyen, Thinh B Nguyen, Sophia Park, Nuz