日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Lysyl-tRNA synthetase, a target for urgently needed M. tuberculosis drugs

赖氨酰-tRNA 合成酶是急需的结核分枝杆菌药物的靶标

Simon R Green, Susan H Davis, Sebastian Damerow, Curtis A Engelhart, Michael Mathieson, Beatriz Baragaña, David A Robinson, Jevgenia Tamjar, Alice Dawson, Fabio K Tamaki, Kirsteen I Buchanan, John Post, Karen Dowers, Sharon M Shepherd, Chimed Jansen, Fabio Zuccotto, Ian H Gilbert, Ola Epemolu, Jenni

Spirocycle MmpL3 Inhibitors with Improved hERG and Cytotoxicity Profiles as Inhibitors of Mycobacterium tuberculosis Growth

具有改进的 hERG 和细胞毒性特征的 Spirocycle MmpL3 抑制剂可作为结核分枝杆菌生长的抑制剂

Peter C Ray, Margaret Huggett, Penelope A Turner, Malcolm Taylor, Laura A T Cleghorn, Julie Early, Anuradha Kumar, Shilah A Bonnett, Lindsay Flint, Douglas Joerss, James Johnson, Aaron Korkegian, Steven Mullen, Abraham L Moure, Susan H Davis, Dinakaran Murugesan, Michael Mathieson, Nicola Caldwell,