日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

In vitro and in vivo characterization of irreversible mutant-selective EGFR inhibitors that are wild-type sparing

不可逆突变选择性 EGFR 抑制剂(保留野生型)的体外和体内表征

Robert Tjin Tham Sjin, Kwangho Lee, Annette O Walter, Aleksandr Dubrovskiy, Michael Sheets, Thia St Martin, Matthew T Labenski, Zhendong Zhu, Richland Tester, Russell Karp, Aravind Medikonda, Prasoon Chaturvedi, Yixuan Ren, Henry Haringsma, Jeff Etter, Mitch Raponi, Andrew D Simmons, Thomas C Hardin

Discovery of a mutant-selective covalent inhibitor of EGFR that overcomes T790M-mediated resistance in NSCLC

发现一种 EGFR 突变选择性共价抑制剂,可克服 NSCLC 中 T790M 介导的耐药性

Annette O Walter, Robert Tjin Tham Sjin, Henry J Haringsma, Kadoaki Ohashi, Jing Sun, Kwangho Lee, Aleksandr Dubrovskiy, Matthew Labenski, Zhendong Zhu, Zhigang Wang, Michael Sheets, Thia St Martin, Russell Karp, Dan van Kalken, Prasoon Chaturvedi, Deqiang Niu, Mariana Nacht, Russell C Petter, Willi

Inhibition of Btk with CC-292 provides early pharmacodynamic assessment of activity in mice and humans

使用 CC-292 抑制 Btk 可对小鼠和人类的活性进行早期药效学评估

Erica K Evans, Richland Tester, Sharon Aslanian, Russell Karp, Michael Sheets, Matthew T Labenski, Steven R Witowski, Heather Lounsbury, Prasoon Chaturvedi, Hormoz Mazdiyasni, Zhendong Zhu, Mariana Nacht, Martin I Freed, Russell C Petter, Alex Dubrovskiy, Juswinder Singh, William F Westlin

Online doctor reviews: do they track surgeon volume, a proxy for quality of care?

在线医生评价:它们是否会追踪外科医生的手术量(手术量是衡量医疗质量的指标)?

Segal, Jeffrey; Sacopulos, Michael; Sheets, Virgil; Thurston, Irish; Brooks, Kendra; Puccia, Ryan