日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Optimized Pyridazinone Nutrient Channel Inhibitors Are Potent and Specific Antimalarial Leads

优化的哒嗪酮营养通道抑制剂是强效且特异的抗疟药物

Michelle M Butler, Samanthi L Waidyarachchi, Jinfeng Shao, Son T Nguyen, Xiaoyuan Ding, Steven C Cardinale, Lucas R Morin, Steven M Kwasny, Mai Ito, Jeanine Gezelle, María B Jiménez-Díaz, Iñigo Angulo-Barturen, Robert T Jacobs, Jeremy N Burrows, Zachary D Aron, Terry L Bowlin, Sanjay A Desai

trans-Translation inhibitors bind to a novel site on the ribosome and clear Neisseria gonorrhoeae in vivo

反式翻译抑制剂与核糖体上的新位点结合,并在体内清除淋病奈瑟菌

Zachary D Aron #, Atousa Mehrani #, Eric D Hoffer #, Kristie L Connolly, Pooja Srinivas, Matthew C Torhan, John N Alumasa, Mynthia Cabrera, Divya Hosangadi, Jay S Barbor, Steven C Cardinale, Steven M Kwasny, Lucas R Morin, Michelle M Butler, Timothy J Opperman, Terry L Bowlin, Ann Jerse, Scott M Sta

MBX-500, a hybrid antibiotic with in vitro and in vivo efficacy against toxigenic Clostridium difficile

MBX-500 是一种混合抗生素,具有体外和体内对抗产毒艰难梭菌的功效

Michelle M Butler, Dean L Shinabarger, Diane M Citron, Ciarán P Kelly, Sofya Dvoskin, George E Wright, Hanping Feng, Saul Tzipori, Terry L Bowlin

Novel Benzimidazole Inhibitors of Botulinum Neurotoxin/A Display Enzyme and Cell-Based Potency

新型苯并咪唑类肉毒杆菌毒素/A 抑制剂展示酶和细胞效力

Steven C Cardinale, Michelle M Butler, Gordon Ruthel, Jonathan E Nuss, Laura M Wanner, Bing Li, Ramdas Pai, Norton P Peet, Sina Bavari, Terry L Bowlin

Comparative in vitro activity profiles of novel bis-indole antibacterials against gram-positive and gram-negative clinical isolates

新型双吲哚抗菌药物对革兰氏阳性菌和革兰氏阴性菌临床分离株的体外活性比较

Michelle M Butler, John D Williams, Norton P Peet, Donald T Moir, Rekha G Panchal, Sina Bavari, Dean L Shinabarger, Terry L Bowlin