日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Integration of the Integrate, Design, Assess, and Share Framework in Developing the Environmental Health Literacy Toolkit Paraben-Free & Me: Protocol for a Randomized Controlled Trial

将“整合、设计、评估和分享”框架应用于环境健康素养工具包的开发;无防腐剂与我:一项随机对照试验方案

De Michino, Graziella; Dhillon, Satveer; Barakat, Caroline

Editor's Note: Small-Molecule Inhibition of the Acyl-Lysine Reader ENL as a Strategy against Acute Myeloid Leukemia

编者按:小分子抑制酰基赖氨酸阅读器ENL作为对抗急性髓系白血病的策略

Liu, Yiman; Li, Qinglan; Alikarami, Fatemeh; Barrett, Declan R; Mahdavi, Leila; Li, Hangpeng; Tang, Sylvia; Khan, Tanweer A; Michino, Mayako; Hill, Connor; Song, Lele; Yang, Lu; Li, Yuanyuan; Pokharel, Sheela Pangeni; Stamford, Andrew W; Liverton, Nigel; Renzetti, Louis M; Taylor, Simon; Watt, Gillian F; Ladduwahetty, Tammy; Kargman, Stacia; Meinke, Peter T; Foley, Michael A; Shi, Junwei; Li, Haitao; Carroll, Martin; Chen, Chun-Wei; Gardini, Alessandro; Maillard, Ivan; Huggins, David J; Bernt, Kathrin M; Wan, Liling

Simulating cell-free chromatin using preclinical cancer models for liquid biopsy applications.

利用临床前癌症模型模拟无细胞染色质,用于液体活检应用。

Main Sasha C, De Michino Steven D, Penny Lucas, Aamir Aleem, Keshavarzian Tina, Lok Benjamin H, Kridel Robert, Cescon David W, Hoffman Michael M, Lupien Mathieu, Bratman Scott V

Discovery of Novel Isofunctional SARS-CoV‑2 NSP14 RNA Cap Methyltransferase Inhibitors by Structure-Based Virtual Screening

通过基于结构的虚拟筛选发现新型同源SARS-CoV-2 NSP14 RNA帽甲基转移酶抑制剂

Meyer, Cindy; Michino, Mayako; Huggins, David J; Garzia, Aitor; Davis, Jada A; Miller, Michael W; Liverton, Nigel; Hoffmann, Hans-Heinrich; Glickman, J Fraser; Nitsche, Julius; Ganichkin, Oleg; Steinbacher, Stefan; Rice, Charles M; Meinke, Peter T; Tuschl, Thomas

Risk perception of personal care products: A scoping review of knowledge translation strategies in environmental health

个人护理产品风险认知:环境健康知识转化策略的范围界定综述

Diyab, Ranim; De Michino, Graziella; Yousufzai, Susan Jamuria; Barakat, Caroline

AI meets physics in computational structure-based drug discovery for GPCRs

人工智能与物理学在基于计算结构的GPCR药物发现中相遇

Michino, Mayako; Vendome, Jeremie; Kufareva, Irina

Indazole to 2-Cyanoindole Scaffold Progression for Mycobacterial Lipoamide Dehydrogenase Inhibitors Achieves Extended Target Residence Time and Improved Antibacterial Activity

吲唑至2-氰基吲哚骨架的合成路线用于制备分枝杆菌硫辛酰胺脱氢酶抑制剂,可延长靶点停留时间并提高抗菌活性。

Sun, Shan; Ginn, John; Kochanczyk, Tomasz; Arango, Nancy; Jiang, Xiuju; Huggins, David J; Bean, James; Michino, Mayako; Baxt, Leigh; Liverton, Nigel; Meinke, Peter T; Bryk, Ruslana

Lead Optimization of Small Molecule ENL YEATS Inhibitors to Enable In Vivo Studies: Discovery of TDI-11055

优化小分子ENL YEATS抑制剂以开展体内研究:TDI-11055的发现

Michino, Mayako; Khan, Tanweer A; Miller, Michael W; Fukase, Yoshiyuki; Vendome, Jeremie; Adura, Carolina; Glickman, J Fraser; Liu, Yiman; Wan, Liling; Allis, C David; Stamford, Andrew W; Meinke, Peter T; Renzetti, Louis M; Kargman, Stacia; Liverton, Nigel J; Huggins, David J

Next-generation neuropeptide Y receptor small-molecule agonists inhibit mosquito-biting behavior

下一代神经肽Y受体小分子激动剂可抑制蚊子叮咬行为

Emely V Zeledon, Leigh A Baxt, Tanweer A Khan, Mayako Michino, Michael Miller, David J Huggins, Caroline S Jiang, Leslie B Vosshall, Laura B Duvall

Next Generation Neuropeptide Y Receptor Small Molecule Agonists Inhibit Mosquito Biting Behavior

下一代神经肽Y受体小分子激动剂抑制蚊子叮咬行为

Emely V Zeledon, Leigh A Baxt, Tanweer A Khan, Mayako Michino, Michael Miller, David J Huggins, Caroline S Jiang, Leslie B Vosshall, Laura B Duvall