日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

QW-5-70 targets the colchicine site and demonstrates antitumor activity in P-gp-overexpressing cancer models

QW-5-70靶向秋水仙碱结合位点,并在P-gp过表达的癌症模型中表现出抗肿瘤活性。

Xie, Yang; Hou, Ruida; Albadari, Najah; Chen, Hao; Miller, Darcie J; Quadrozzi Gruntz, Judith; Oldham, Michael L; Kamal, Mir Shahriar; Jiang, Jianxiong; Wu, Zhongzhi; Miller, Duane D; Li, Wei

VERU-111 Promotes an Anti-Tumor Response Through Restoration of Gut Microbial Homeostasis and Associated Metabolic Dysregulation

VERU-111通过恢复肠道微生物稳态和相关的代谢紊乱来促进抗肿瘤反应

Mamun, Md Abdullah Al; Rakib, Ahmed; Mandal, Mousumi; Li, Wei; Miller, Duane D; Chen, Hao; Nagarkatti, Mitzi; Nagarkatti, Prakash; Singh, Udai P

Design and synthesis of novel 4-aryl-2-benzoyl-imidazoles as colchicine binding site inhibitors.

设计和合成新型 4-芳基-2-苯甲酰基咪唑类化合物作为秋水仙碱结合位点抑制剂

Albadari Najah, Xie Yang, Wang Qinghui, Miller Darcie J, Gruntz Judith Quadrozzi, Oldham Michael L, Chen Hao, Ma Dejian, Wu Zhongzhi, Miller Duane D, Li Wei

Discovery of potent and brain-penetrable tubulin inhibitors that effectively suppress breast cancer brain metastasis.

发现强效且能穿透血脑屏障的微管蛋白抑制剂,可有效抑制乳腺癌脑转移。

Krutilina Raisa I, Adeleye Kelli L, Playa Hilaire C, Pochampally Satyanarayana, Banjeree Souvik, Oluwalana Damilola, Kamal Mir Shahriar, Tian Di, Miller Duane D, Li Wei, Seagroves Tiffany N

Structural Activity Relationship Analysis of New Diphenyl PFI-3 Analogues Targeting for the Treatment of Glioblastoma

针对胶质母细胞瘤治疗的新型二苯基PFI-3类似物的结构活性关系分析

Hwang, Dong-Jin; Yang, Chuanhe; Wang, Yinan; Kelso, Hannah; Pochampally, Satyanarayana; Pfeffer, Lawrence M; Miller, Duane D

A Pyrimidine-Based Tubulin Inhibitor Shows Potent Anti-Glioblastoma Activity In Vitro and In Vivo

一种基于嘧啶的微管蛋白抑制剂在体外和体内均显示出强大的抗胶质母细胞瘤活性

Pochampally, Satyanarayana; Pfeffer, Lawrence M; Miranda-Carboni, Gustavo A; Daniel, Macey; James, Jazz I; Smith, Allana; Yang, Chuan He; Kelso, Hannah R; Parke, Deanna N; Hwang, Dong-Jin; Li, Wei; Miller, Duane D

Tyr1497 in the BRG1 Bromodomain of the SWI/SNF Complex is Critical for the Binding and Function of a Selective BRG1 Inhibitor

SWI/SNF复合物BRG1溴结构域中的Tyr1497对于选择性BRG1抑制剂的结合和功能至关重要

Wang, Yinan; Yang, Chuanhe; Miranda-Carboni, Gustavo A; Kelso, Hannah; Seetharaman, Jayaraman; Hwang, Dong-Jin; Miller, Duane D; Pfeffer, Lawrence M

Discovery of a potent and selective TRPC3 antagonist with neuroprotective effects.

发现了一种具有神经保护作用的强效选择性 TRPC3 拮抗剂

Wang Jiaxing, Zhang Sicheng, Boda Vijay K, Chen Hao, Park Hyunseo, Parmar Keyur, Ma Dejian, Miller Duane D, Meibohm Bernd, Du Jianyang, Liao Francesca-Fang, Wu Zhongzhi, Li Wei

Biological activity of a stable 6-aryl-2-benzoyl-pyridine colchicine-binding site inhibitor, 60c, in metastatic, triple-negative breast cancer.

稳定的 6-芳基-2-苯甲酰基-吡啶秋水仙碱结合位点抑制剂 60c 在转移性三阴性乳腺癌中的生物活性

Oluwalana Damilola, Adeleye Kelli L, Krutilina Raisa I, Chen Hao, Playa Hilaire, Deng Shanshan, Parke Deanna N, Abernathy John, Middleton Leona, Cullom Alexandra, Thalluri Bhargavi, Ma Dejian, Meibohm Bernd, Miller Duane D, Seagroves Tiffany N, Li Wei

A molecular switch from tumor suppressor to oncogene in ER+ve breast cancer: Role of androgen receptor, JAK-STAT, and lineage plasticity

ER阳性乳腺癌中肿瘤抑制基因向癌基因的分子转换:雄激素受体、JAK-STAT和谱系可塑性的作用

Asemota, Sarah; Effah, Wendy; Holt, Jeremiah; Johnson, Daniel; Cripe, Linnea; Ponnusamy, Suriyan; Thiyagarajan, Thirumagal; Khosrosereshki, Yekta; Hwang, Dong-Jin; He, Yali; Grimes, Brandy; Fleming, Martin D; Pritchard, Frances E; Hendrix, Ashley; Fan, Meiyun; Jain, Abhinav; Choi, Hyo Young; Makowski, Liza; Hayes, D Neil; Miller, Duane D; Pfeffer, Lawrence M; Santhanam, Balaji; Narayanan, Ramesh