日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Intracrine FFA4 signaling controls lipolysis at lipid droplets.

细胞内 FFA4 信号传导控制脂滴处的脂肪分解。

O'Brien Shannon L, Tripp Emma, Barki Natasja, Blondel-Tepaz Elodie, Smith Gabrielle, Boufersaoui Adam, Roberts Jennie, Pike Jeremy A, Correia Joao, Miljus Tamara, Bouvier Michel, Tennant Daniel A, Hudson Brian D, Gerhart-Hines Zachary, Milligan Graeme, Schwartz Thue W, Calebiro Davide

Shaping Antimalarials: A Geometry-First Approach to PfCLK3 Covalent Inhibitors

抗疟药的调控:一种基于几何结构的PfCLK3共价抑制剂设计方法

Brettell, Skye B; Fuentes-Guerra Bustos, Carla; Sharma, Saumya; Cann, Gillian; Carruthers, Lauren V; Begen, Abbey; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Discovery, Structure-Activity Relationship, and Functional Characterization of a Chromenopyrrole Series as Orthosteric Antagonists of GPR84

色烯吡咯系列化合物作为GPR84正构拮抗剂的发现、构效关系及功能表征

Malone, Michael A; Yin, Ruijing; Li, Yueming; Jenkins, Laura; Guseinov, Abdul-Akim; Marsango, Sara; Huggett, Mark; Huggett, Margaret; Boyle, Anna; Morrison, Angus; Tikhonova, Irina G; Milligan, Graeme; Jamieson, Andrew G

Steroid Recognition in Adhesion GPCRs: A Structural and Pharmacological Perspective

粘附 GPCR 中的类固醇识别:结构和药理学视角

Fleming, Bethany; Guseinov, Abdul-Akim; Tikhonova, Irina G; Milligan, Graeme; Perry-Hauser, Nicole A

Mechanism of GPR84 allosteric modulation at a helix 8-proximate site

GPR84 在螺旋 8 近端位点的变构调节机制

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Zhou, Jingkai; Gossen, Fabian; Wang, Pinqi; Al Mahmud, Zobaer; Li, Yueming; Mahardhika, Andhika B; Muller, Christa E; Feng, Mingye; Russell, Angela J; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

Allosteric modulation and biased signalling at free fatty acid receptor 2

游离脂肪酸受体 2 的变构调节和偏向性信号传导

Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; Valentini, Alice; Marsango, Sara; Schultz-Knudsen, Katrine; Ulven, Trond; Rexen Ulven, Elisabeth; Tikhonova, Irina G; Milligan, Graeme; Zhang, Cheng

NaBC1 Boron Transporter Enables Myoblast Response to Substrate Rigidity via Fibronectin-Binding Integrins.

NaBC1 硼转运蛋白通过纤连蛋白结合整合素使成肌细胞对底物刚性做出反应

Gonzalez-Valdivieso Juan, Ciccone Giuseppe, Dhawan Udesh, Quon Tezz, Barcelona-Estaje Eva, Rodrigo-Navarro Aleixandre, Castillo Rafael R, Milligan Graeme, Rico Patricia, Salmeron-Sanchez Manuel

G Protein-Coupled Receptor 35 Suppresses Oxidative Stress Responsive Kinase 1 in Diabetic Wound Healing.

G蛋白偶联受体35抑制糖尿病伤口愈合中的氧化应激反应激酶1

Li Hainan, Xu Liping, Meda Venkata Sai Pranathi, Minjares Morgan, Melhem Hassan, Kowluru Anjaneyulu, Niess Jan Hendrik, Milligan Graeme, Wang Jie-Mei

Lysine targeting covalent inhibitors of malarial kinase PfCLK3

赖氨酸靶向共价抑制疟原虫激酶 PfCLK3 的抑制剂

Brettell, Skye B; Cann, Gillian; Begen, Abbey; Sharma, Saumya; Mahindra, Amit; Carruthers, Lauren V; Milligan, Graeme; Clarke, David J; Tobin, Andrew B; Jamieson, Andrew G

Steric control of signaling bias in the immunometabolic receptor GPR84

免疫代谢受体 GPR84 中信号偏向的空间控制

Wang, Pinqi; Zhang, Xuan; Guseinov, Abdul-Akim; Jenkins, Laura; von Hallerstein, Carl; Colburn, Jonathan D; Ives, Rowan; Luscombe, Vincent B; Marsango, Sara; Oktavia, Listiana; Raja, Arun; Greaves, David R; Biggin, Philip C; Milligan, Graeme; Zhang, Cheng; Tikhonova, Irina G; Russell, Angela J