日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polypharmacology of an Optimal Kinase Library

最优激酶库的多药理学

Mills, Caitlin E; Hug, Clemens; Sajeevan, Karuna Anna; Clark, Nicholas; Victor, Chiara; Chung, Mirra; Rawat, Sameer; Aldridge, Bree; Albers, Mark W; Chowdhury, Ratul; Gyori, Benjamin M; Sorger, Peter K

Corrigendum to "Comprehensive Proteomics Metadata and Integrative Web Portals Facilitate Sharing and Integration of LINCS Multiomics Data"

关于“综合蛋白质组学元数据和集成网络门户促进LINCS多组学数据的共享和整合”一文的更正

Vidović, Dušica; Shamsaei, Behrouz; Schürer, Stephan C; Kogan, Phillip; Chojnacki, Szymon; Kouril, Michal; Medvedovic, Mario; Niu, Wen; Azeloglu, Evren U; Birtwistle, Marc R; Chen, Yibang; Chen, Tong; Hansen, Jens; Hu, Bin; Iyengar, Ravi; Jayaraman, Gomathi; Li, Hong; Liu, Tong; Sobie, Eric A; Xiong, Yuguang; Berberich, Matthew J; Bradshaw, Gary; Chung, Mirra; Everley, Robert A; Gaudio, Ben; Hafner, Marc; Kalocsay, Marian; Mills, Caitlin E; Nariya, Maulik K; Sorger, Peter K; Subramanian, Kartik; Victor, Chiara; Banuelos, Maria; Dardov, Victoria; Holewinski, Ronald; Manalo, Danica-Mae; Mandefro, Berhan; Matlock, Andrea D; Ornelas, Loren; Sareen, Dhruv; Svendsen, Clive N; Vaibhav, Vineet; Van Eyk, Jennifer E; Venkatraman, Vidya; Finkbiener, Steve; Fraenkel, Ernest; Rothstein, Jeffrey; Thompson, Leslie; Asiedu, Jacob; Carr, Steven A; Christianson, Karen E; Davison, Desiree; Dele-Oni, Deborah O; DeRuff, Katherine C; Egri, Shawn B; Vaca Jacome, Alvaro Sebastian; Jaffe, Jacob D; Lam, Daniel; Litichevskiy, Lev; Lu, Xiaodong; Mullahoo, James; Officer, Adam; Papanastasiou, Malvina; Peckner, Ryan; Toder, Caidin; Blanchard, Joel; Bula, Michael; Ko, Tak; Tsai, Li-Huei; Young, Jennie Z; Sharma, Vagisha; Meller, Jarek; MacCoss, Michael J

Comprehensive Proteomics Metadata and Integrative Web Portals Facilitate Sharing and Integration of LINCS Multiomics Data

全面的蛋白质组学元数据和集成式网络门户促进了LINCS多组学数据的共享和整合。

Vidović, Dušica; Shamsaei, Behrouz; Schürer, Stephan C; Kogan, Phillip; Chojnacki, Szymon; Kouril, Michal; Medvedovic, Mario; Niu, Wen; Azeloglu, Evren U; Birtwistle, Marc R; Chen, Yibang; Chen, Tong; Hansen, Jens; Hu, Bin; Iyengar, Ravi; Jayaraman, Gomathi; Li, Hong; Liu, Tong; Sobie, Eric A; Xiong, Yuguang; Berberich, Matthew J; Bradshaw, Gary; Chung, Mirra; Everley, Robert A; Gaudio, Ben; Hafner, Marc; Kalocsay, Marian; Mills, Caitlin E; Nariya, Maulik K; Sorger, Peter K; Subramanian, Kartik; Victor, Chiara; Banuelos, Maria; Dardov, Victoria; Holewinski, Ronald; Manalo, Danica-Mae; Mandefro, Berhan; Matlock, Andrea D; Ornelas, Loren; Sareen, Dhruv; Svendsen, Clive N; Vaibhav, Vineet; Van Eyk, Jennifer E; Venkatraman, Vidya; Finkbiener, Steve; Fraenkel, Ernest; Rothstein, Jeffrey; Thompson, Leslie; Asiedu, Jacob; Carr, Steven A; Christianson, Karen E; Davison, Desiree; Dele-Oni, Deborah O; DeRuff, Katherine C; Egri, Shawn B; Jacome, Alvaro Sebastian Vaca; Jaffe, Jacob D; Lam, Daniel; Litichevskiy, Lev; Lu, Xiaodong; Mullahoo, James; Officer, Adam; Papanastasiou, Malvina; Peckner, Ryan; Toder, Caidin; Blanchard, Joel; Bula, Michael; Ko, Tak; Tsai, Li-Huei; Young, Jennie Z; Sharma, Vagisha; Pillai, Ajay; Meller, Jarek; MacCoss, Michael J

Discovery of bivalent small molecule degraders of cyclin-dependent kinase 7 (CDK7).

发现细胞周期蛋白依赖性激酶 7 (CDK7) 的二价小分子降解剂

Ji Wenzhi, Du Guangyan, Jiang Jie, Lu Wenchao, Mills Caitlin E, Yuan Linjie, Jiang Fen, He Zhixiang, Bradshaw Gary A, Chung Mirra, Jiang Zixuan, Byun Woong Sub, Hinshaw Stephen M, Zhang Tinghu, Gray Nathanael S

Paired evaluation of machine-learning models characterizes effects of confounders and outliers

机器学习模型的配对评估可以表征混杂因素和异常值的影响。

Nariya, Maulik K; Mills, Caitlin E; Sorger, Peter K; Sokolov, Artem

The Kinase Chemogenomic Set (KCGS): An Open Science Resource for Kinase Vulnerability Identification

激酶化学基因组学数据集(KCGS):用于识别激酶脆弱性的开放科学资源

Wells, Carrow I; Al-Ali, Hassan; Andrews, David M; Asquith, Christopher R M; Axtman, Alison D; Dikic, Ivan; Ebner, Daniel; Ettmayer, Peter; Fischer, Christian; Frederiksen, Mathias; Futrell, Robert E; Gray, Nathanael S; Hatch, Stephanie B; Knapp, Stefan; Lücking, Ulrich; Michaelides, Michael; Mills, Caitlin E; Müller, Susanne; Owen, Dafydd; Picado, Alfredo; Saikatendu, Kumar S; Schröder, Martin; Stolz, Alexandra; Tellechea, Mariana; Turunen, Brandon J; Vilar, Santiago; Wang, Jinhua; Zuercher, William J; Willson, Timothy M; Drewry, David H

Development of CDK2 and CDK5 Dual Degrader TMX-2172

CDK2 和 CDK5 双重降解剂 TMX-2172 的开发

Teng, Mingxing; Jiang, Jie; He, Zhixiang; Kwiatkowski, Nicholas P; Donovan, Katherine A; Mills, Caitlin E; Victor, Chiara; Hatcher, John M; Fischer, Eric S; Sorger, Peter K; Zhang, Tinghu; Gray, Nathanael S

The Library of Integrated Network-Based Cellular Signatures NIH Program: System-Level Cataloging of Human Cells Response to Perturbations

美国国立卫生研究院(NIH)项目“基于网络的细胞特征库”:人类细胞对扰动反应的系统级编目

Keenan, Alexandra B; Jenkins, Sherry L; Jagodnik, Kathleen M; Koplev, Simon; He, Edward; Torre, Denis; Wang, Zichen; Dohlman, Anders B; Silverstein, Moshe C; Lachmann, Alexander; Kuleshov, Maxim V; Ma'ayan, Avi; Stathias, Vasileios; Terryn, Raymond; Cooper, Daniel; Forlin, Michele; Koleti, Amar; Vidovic, Dusica; Chung, Caty; Schürer, Stephan C; Vasiliauskas, Jouzas; Pilarczyk, Marcin; Shamsaei, Behrouz; Fazel, Mehdi; Ren, Yan; Niu, Wen; Clark, Nicholas A; White, Shana; Mahi, Naim; Zhang, Lixia; Kouril, Michal; Reichard, John F; Sivaganesan, Siva; Medvedovic, Mario; Meller, Jaroslaw; Koch, Rick J; Birtwistle, Marc R; Iyengar, Ravi; Sobie, Eric A; Azeloglu, Evren U; Kaye, Julia; Osterloh, Jeannette; Haston, Kelly; Kalra, Jaslin; Finkbiener, Steve; Li, Jonathan; Milani, Pamela; Adam, Miriam; Escalante-Chong, Renan; Sachs, Karen; Lenail, Alex; Ramamoorthy, Divya; Fraenkel, Ernest; Daigle, Gavin; Hussain, Uzma; Coye, Alyssa; Rothstein, Jeffrey; Sareen, Dhruv; Ornelas, Loren; Banuelos, Maria; Mandefro, Berhan; Ho, Ritchie; Svendsen, Clive N; Lim, Ryan G; Stocksdale, Jennifer; Casale, Malcolm S; Thompson, Terri G; Wu, Jie; Thompson, Leslie M; Dardov, Victoria; Venkatraman, Vidya; Matlock, Andrea; Van Eyk, Jennifer E; Jaffe, Jacob D; Papanastasiou, Malvina; Subramanian, Aravind; Golub, Todd R; Erickson, Sean D; Fallahi-Sichani, Mohammad; Hafner, Marc; Gray, Nathanael S; Lin, Jia-Ren; Mills, Caitlin E; Muhlich, Jeremy L; Niepel, Mario; Shamu, Caroline E; Williams, Elizabeth H; Wrobel, David; Sorger, Peter K; Heiser, Laura M; Gray, Joe W; Korkola, James E; Mills, Gordon B; LaBarge, Mark; Feiler, Heidi S; Dane, Mark A; Bucher, Elmar; Nederlof, Michel; Sudar, Damir; Gross, Sean; Kilburn, David F; Smith, Rebecca; Devlin, Kaylyn; Margolis, Ron; Derr, Leslie; Lee, Albert; Pillai, Ajay