日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Enhanced contrast in FAP-targeting PET imaging with (61)Cu-labeled FAP inhibitors: development and preclinical evaluation of novel [(61)Cu]Cu-Kalios PET radioligands

利用 (61)Cu 标记的 FAP 抑制剂增强 FAP 靶向 PET 成像的对比度:新型 [(61)Cu]Cu-Kalios PET 放射性配体的开发和临床前评估

Millul, Jacopo; Basaco Bernabeu, Tais; Gaonkar, Raghuvir H; De Rose, Francesco; Jaafar-Thiel, Leila; Ulaner, Gary A; Mansi, Rosalba; Fani, Melpomeni

Head-to-head comparison of different classes of FAP radioligands designed to increase tumor residence time: monomer, dimer, albumin binders, and small molecules vs peptides

不同类型FAP放射性配体(旨在延长肿瘤停留时间)的直接比较:单体、二聚体、白蛋白结合剂和小分子与肽类

Millul, Jacopo; Koepke, Lennart; Haridas, Gaonkar Raghuvir; Sparrer, Konstantin M J; Mansi, Rosalba; Fani, Melpomeni

Translational imaging of the fibroblast activation protein (FAP) using the new ligand [(68)Ga]Ga-OncoFAP-DOTAGA

利用新型配体[(68)Ga]Ga-OncoFAP-DOTAGA对成纤维细胞活化蛋白(FAP)进行转化成像

Backhaus, P; Gierse, F; Burg, M C; Büther, F; Asmus, I; Dorten, P; Cufe, J; Roll, W; Neri, D; Cazzamalli, S; Millul, J; Mock, J; Galbiati, A; Zana, A; Schäfers, K P; Hermann, S; Weckesser, M; Tio, J; Wagner, S; Breyholz, H-J; Schäfers, M

Automated Radiosynthesis, Preliminary In Vitro/In Vivo Characterization of OncoFAP-Based Radiopharmaceuticals for Cancer Imaging and Therapy

基于OncoFAP的放射性药物在癌症成像和治疗中的自动化放射合成、初步体外/体内表征

Bartoli, Francesco; Elsinga, Philip; Nazario, Luiza Reali; Zana, Aureliano; Galbiati, Andrea; Millul, Jacopo; Migliorini, Francesca; Cazzamalli, Samuele; Neri, Dario; Slart, Riemer H J A; Erba, Paola Anna

A Dimeric FAP-Targeting Small-Molecule Radioconjugate with High and Prolonged Tumor Uptake

一种靶向FAP的二聚体小分子放射性偶联物,具有高且持久的肿瘤摄取

Galbiati, Andrea; Zana, Aureliano; Bocci, Matilde; Millul, Jacopo; Elsayed, Abdullah; Mock, Jacqueline; Neri, Dario; Cazzamalli, Samuele

Stereo- and regiodefined DNA-encoded chemical libraries enable efficient tumour-targeting applications

立体选择性和区域选择性明确的DNA编码化学库能够实现高效的肿瘤靶向应用

Favalli, Nicholas; Bassi, Gabriele; Pellegrino, Christian; Millul, Jacopo; De Luca, Roberto; Cazzamalli, Samuele; Yang, Su; Trenner, Anika; Mozaffari, Nour L; Myburgh, Renier; Moroglu, Mustafa; Conway, Stuart J; Sartori, Alessandro A; Manz, Markus G; Lerner, Richard A; Vogt, Peter K; Scheuermann, Jörg; Neri, Dario

An ultra-high-affinity small organic ligand of fibroblast activation protein for tumor-targeting applications.

一种对成纤维细胞激活蛋白具有超高亲和力的小分子有机配体,可用于肿瘤靶向治疗

Millul Jacopo, Bassi Gabriele, Mock Jacqueline, Elsayed Abdullah, Pellegrino Christian, Zana Aureliano, Dakhel Plaza Sheila, Nadal Lisa, Gloger Andreas, Schmidt Eleonore, Biancofiore Ilaria, Donckele Etienne J, Samain Florent, Neri Dario, Cazzamalli Samuele

Immunotherapy with Immunocytokines and PD-1 Blockade Enhances the Anticancer Activity of Small Molecule-Drug Conjugates Targeting Carbonic Anhydrase IX

免疫细胞因子和PD-1阻断联合免疫疗法可增强靶向碳酸酐酶IX的小分子药物偶联物的抗癌活性

Millul, Jacopo; Krudewig, Christiane; Zana, Aureliano; Dakhel Plaza, Sheila; Puca, Emanuele; Villa, Alessandra; Neri, Dario; Cazzamalli, Samuele

Sortase-Mediated Site-Specific Modification of Interleukin-2 for the Generation of a Tumor-Targeting Acetazolamide-Cytokine Conjugate

分选酶介导的白细胞介素-2 位点特异性修饰用于生成肿瘤靶向乙酰唑胺-细胞因子缀合物

Baptiste Gouyou, Jacopo Millul, Alessandra Villa, Samuele Cazzamalli, Dario Neri, Mattia Matasci

Design and conduct of the activated protein C and corticosteroids for human septic shock (APROCCHSS) trial

设计和实施活化蛋白C和皮质类固醇治疗人类脓毒性休克(APROCCHSS)试验

Annane, Djillali; Buisson, Christian Brun; Cariou, Alain; Martin, Claude; Misset, Benoit; Renault, Alain; Lehmann, Blandine; Millul, Valérie; Maxime, Virginie; Bellissant, Eric