日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mimicking Nature in Reshaping the Triterpene Skeleton: Synthesis of a Class of Unnatural Oleanane Derivatives

模仿自然重塑三萜骨架:一类非天然齐墩果烷衍生物的合成

di Biase, Edoardo; Gargiulo, Ernesto; Imperio, Daniela; Chianese, Giuseppina; Caprioglio, Diego; Amin, Hawraz Ibrahim M; Taglialatela-Scafati, Orazio; Minassi, Alberto

The Impact of a Quinone Scaffold on Thermo-TRPs Modulation by Dimethylheptyl Phytocannabinoids

醌骨架对二甲基庚基植物大麻素调节热致色氨酸受体的影响

Schiano Moriello, Aniello; Bossoni, Aurora; Mattoteia, Daiana; Caprioglio, Diego; Minassi, Alberto; Appendino, Giovanni; De Petrocellis, Luciano; Amodeo, Pietro; Vitale, Rosa Maria

Optimization of Steroid Photochemistry and Its Application in the Synthesis of 5,6-Dihydro-Ophiopogonol A

类固醇光化学的优化及其在5,6-二氢麦冬酚A合成中的应用

Maioli, Chiara; Lauro, Gianluigi; Sategna, Anna; Caprioglio, Diego; Amin, Hawraz Ibrahim M; D'Auria, Maurizio; Imperio, Daniela; Bifulco, Giuseppe; Minassi, Alberto

Stereoselective Shi-type epoxidation with 3-oxo-4,6-O-benzylidene pyranoside catalysts: unveiling the role of carbohydrate skeletons

利用3-氧代-4,6-O-亚苄基吡喃糖苷催化剂进行立体选择性Shi型环氧化反应:揭示碳水化合物骨架的作用

Imperio, Daniela; Valloni, Filippo; Caprioglio, Diego; Minassi, Alberto; Casali, Emanuele; Panza, Luigi

The synthetic triterpenoids CDDO-TFEA and CDDO-Me, but not CDDO, promote nuclear exclusion of BACH1 impairing its activity

合成三萜类化合物 CDDO-TFEA 和 CDDO-Me(而非 CDDO)可促进 BACH1 的核排斥,从而损害其活性

Laura Casares, Rita Moreno, Kevin X Ali, Maureen Higgins, Sharadha Dayalan Naidu, Graham Neill, Lena Cassin, Anders E Kiib, Esben B Svenningsen, Alberto Minassi, Tadashi Honda, Thomas B Poulsen, Clotilde Wiel, Volkan I Sayin, Albena T Dinkova-Kostova, David Olagnier, Laureano de la Vega

Curcumin-based-fluorescent probes targeting ALDH1A3 as a promising tool for glioblastoma precision surgery and early diagnosis

以 ALDH1A3 为靶点的姜黄素荧光探针有望成为胶质母细胞瘤精准手术和早期诊断的有力工具

Edoardo L M Gelardi #, Diego Caprioglio #, Giorgia Colombo, Erika Del Grosso, Daniele Mazzoletti, Daiana Mattoteia, Stefano Salamone, Davide M Ferraris, Eleonora Aronica, Giulia Nato, Annalisa Buffo, Menico Rizzi, Lorenzo Magrassi, Alberto Minassi, Silvia Garavaglia

Pyrazole-Curcumin Suppresses Cardiomyocyte Hypertrophy by Disrupting the CDK9/CyclinT1 Complex

吡唑-姜黄素通过破坏 CDK9/CyclinT1 复合物抑制心肌细胞肥大

Masafumi Funamoto, Yoichi Sunagawa, Mai Gempei, Kana Shimizu, Yasufumi Katanasaka, Satoshi Shimizu, Toshihide Hamabe-Horiike, Giovanni Appendino, Alberto Minassi, Andreas Koeberle, Maki Komiyama, Kiyoshi Mori, Koji Hasegawa, Tatsuya Morimoto

First thermostable CLIP- tag by rational design applied to an archaeal O6 -alkyl-guanine-DNA-alkyl-transferase

第一个经过合理设计的耐热 CLIP 标签应用于古细菌 O6-烷基鸟嘌呤-DNA-烷基转移酶

Rosa Merlo, Rosanna Mattossovich, Marianna Genta, Anna Valenti, Giovanni Di Mauro, Alberto Minassi, Riccardo Miggiano, Giuseppe Perugino

Cannabinol: History, Syntheses, and Biological Profile of the Greatest "Minor" Cannabinoid

大麻酚:最伟大的“次要”大麻素的历史、合成和生物学特性

Maioli, Chiara; Mattoteia, Daiana; Amin, Hawraz Ibrahim M; Minassi, Alberto; Caprioglio, Diego

Identification of a Novel Curcumin Derivative Influencing Notch Pathway and DNA Damage as a Potential Therapeutic Agent in T-ALL

鉴定出一种影响 Notch 通路和 DNA 损伤的新型姜黄素衍生物作为 T-ALL 的潜在治疗剂

Nadezda Zhdanovskaya, Sara Lazzari, Diego Caprioglio, Mariarosaria Firrincieli, Chiara Maioli, Eleonora Pace, Daniela Imperio, Claudio Talora, Diana Bellavia, Saula Checquolo, Mattia Mori, Isabella Screpanti, Alberto Minassi, Rocco Palermo