A Selective and Orally Bioavailable Quinoline-6-Carbonitrile-Based Inhibitor of CDK8/19 Mediator Kinase with Tumor-Enriched Pharmacokinetics
一种选择性强、口服生物利用度高的喹啉-6-腈基 CDK8/19 介导激酶抑制剂,具有肿瘤富集药代动力学特征
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c01951
Zhang, Li; Cheng, Chen; Li, Jing; Wang, Lili; Chumanevich, Alexander A; Porter, Donald C; Mindich, Aleksei; Gorbunova, Svetlana; Roninson, Igor B; Chen, Mengqian; McInnes, Campbell