日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Light-Driven Organocatalytic Birch Reduction for Late-Stage Drug Modification and sp(3)-Rich Spirocycle Synthesis

光驱动有机催化桦木还原反应用于药物后期修饰和富含sp(3)杂化碳的螺环化合物合成

Schiel, Florian; di Martile, Luca; Coccia, Roberta; Palone, Andrea; Medrzycka, Magdalena; Kqiku, Laura; Neves, Paulo; Matera, Nunzio; Misale, Antonio; Melchiorre, Paolo

Direct Inhibition of RAS Reveals the Features of Oncogenic Signaling Driven by RAS G12 and Q61 Mutations.

直接抑制 RAS 揭示了由 RAS G12 和 Q61 突变驱动的致癌信号的特征

Marasco Michelangelo, Kumar Dinesh, Garcia Borrego Santiago, Seale Tessa, Maddalena Giulia, Mezzadra Riccardo, Belanger Kylie, Cole Soren, Perez Brayan, Luan Wei, Mukherjee Radha, Aricescu Ilinca, Markov Vladimir, Zhu Yuxin, Arena Sabrina, Bardelli Alberto, de Stanchina Elisa, Lowe Scott W, Burkhart Richard A, Zimmerman Jacquelyn W, Yaeger Rona, Kopetz Scott E, Rosen Neal, Misale Sandra

Concurrent SOS1 and MEK suppression inhibits signaling and growth of NF1-null melanoma

同时抑制SOS1和MEK可抑制NF1缺失型黑色素瘤的信号传导和生长。

Michelangelo Marasco ,Dinesh Kumar ,Tessa Seale ,Santiago Garcia Borrego ,Esther Kaplun ,Ilinca Aricescu ,Soren Cole ,Besnik Qeriqi ,Juan Qiu ,Xiaoping Chen ,Amber Bahr ,Deborah Fidele ,Marco H Hofmann ,Daniel Gerlach ,Fabio Savarese ,Taha Merghoub ,Jedd D Wolchok ,Zhan Yao ,Elisa de Stanchina ,David Solit ,Sandra Misale ,Neal Rosen

EGFR-directed antibodies promote HER2 ADC internalization and efficacy

EGFR靶向抗体促进HER2 ADC内化并提高疗效

Avantika Gupta,Flavia Michelini,Hong Shao,Celine Yeh,Joshua Z Drago,Dazhi Liu,Eric Rosiek,Yevgeniy Romin,Negin Ghafourian,Sheeno Thyparambil,Sandra Misale,Wungki Park,Elisa de Stanchina,Yelena Y Janjigian,Rona Yaeger,Bob T Li,Sarat Chandarlapaty

Combined RAF and MEK Inhibition to Treat Activated Non-V600 BRAF-Altered Advanced Cancers

RAF 和 MEK 联合抑制治疗活化的非 V600 BRAF 变异晚期癌症

Naryan Rustgi, Ann Maria, Nicolas Toumbacaris, HuiYong Zhao, Katherine Kargus, Morgan Bryant, Alexandra Waksmundzki, Ilinca Aricescu, Robert A Lefkowitz, Bob T Li, Joanne Chou, Marinela Capanu, Elisa de Stanchina, Sandra Misale, Jinru Shia, Rona Yaeger

Catalytic undirected borylation of tertiary C-H bonds in bicyclo[1.1.1]pentanes and bicyclo[2.1.1]hexanes

双环[1.1.1]戊烷和双环[2.1.1]己烷中叔碳氢键的催化非定向硼化反应

Yu, Isaac F; Manske, Jenna L; Diéguez-Vázquez, Alejandro; Misale, Antonio; Pashenko, Alexander E; Mykhailiuk, Pavel K; Ryabukhin, Sergey V; Volochnyuk, Dmitriy M; Hartwig, John F

Anatomic position determines oncogenic specificity in melanoma

解剖位置决定黑色素瘤的致癌特异性

Joshua M Weiss, Miranda V Hunter, Nelly M Cruz, Arianna Baggiolini, Mohita Tagore, Yilun Ma, Sandra Misale, Michelangelo Marasco, Theresa Simon-Vermot, Nathaniel R Campbell, Felicity Newell, James S Wilmott, Peter A Johansson, John F Thompson, Georgina V Long, John V Pearson, Graham J Mann, Richard

Expanding the Reach of Precision Oncology by Drugging All KRAS Mutants

通过对所有 KRAS 突变体进行药物治疗来扩大精准肿瘤学的应用范围

Hofmann, Marco H; Gerlach, Daniel; Misale, Sandra; Petronczki, Mark; Kraut, Norbert

KRAS (G12C) Mutation Is Associated with Increased Risk of Recurrence in Surgically Resected Lung Adenocarcinoma

KRAS (G12C) 突变与手术切除的肺腺癌复发风险增加相关

Jones, Gregory D; Caso, Raul; Tan, Kay See; Mastrogiacomo, Brooke; Sanchez-Vega, Francisco; Liu, Yuan; Connolly, James G; Murciano-Goroff, Yonina R; Bott, Matthew J; Adusumilli, Prasad S; Molena, Daniela; Rocco, Gaetano; Rusch, Valerie W; Sihag, Smita; Misale, Sandra; Yaeger, Rona; Drilon, Alexander; Arbour, Kathryn C; Riely, Gregory J; Rosen, Neal; Lito, Piro; Zhang, Haiying; Lyden, David C; Rudin, Charles M; Jones, David R; Li, Bob T; Isbell, James M

Post-traumatic peripheral vestibular disorders (excluding positional vertigo) in workers following head injury

头部损伤后工人创伤后周围性前庭功能障碍(不包括位置性眩晕)

Misale, Priyanka; Hassannia, Fatemeh; Dabiri, Sasan; Brandstaetter, Tom; Rutka, John