日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Designer molecules of the synaptic organizer MDGA1 reveal 3D conformational control of biological function

突触组织者 MDGA1 的设计分子揭示了生物功能的 3D 构象控制

Hubert Lee, Nicolas Chofflet, Jianfang Liu, Shanghua Fan, Zhuoyang Lu, Martin Resua Rojas, Patrick Penndorf, Aaron O Bailey, William K Russell, Mischa Machius, Gang Ren, Hideto Takahashi, Gabby Rudenko

Interplay between hevin, SPARC, and MDGAs: Modulators of neurexin-neuroligin transsynaptic bridges

Hevin、SPARC 和 MDGA 之间的相互作用:神经连接蛋白-神经胶质蛋白跨突触桥的调节剂

Shanghua Fan, Shanti Pal Gangwar, Mischa Machius, Gabby Rudenko

Highly Conserved Molecular Features in IgLONs Contrast Their Distinct Structural and Biological Outcomes

IgLON 中高度保守的分子特征与其独特的结构和生物学结果形成对比

Harikanth Venkannagari, James M Kasper, Anurag Misra, Scott A Rush, Shanghua Fan, Hubert Lee, Hong Sun, Suchithra Seshadrinathan, Mischa Machius, Jonathan D Hommel, Gabby Rudenko

Self-assembly of the bZIP transcription factor ΔFosB

bZIP 转录因子 ΔFosB 的自组装

Zhou Yin, Harikanth Venkannagari, Haley Lynch, Galina Aglyamova, Mukund Bhandari, Mischa Machius, Eric J Nestler, Alfred J Robison, Gabby Rudenko

Activator Protein-1: redox switch controlling structure and DNA-binding

激活蛋白-1:氧化还原开关控制结构和 DNA 结合

Zhou Yin, Mischa Machius, Eric J Nestler, Gabby Rudenko

TIR-only protein RBA1 recognizes a pathogen effector to regulate cell death in Arabidopsis

TIR 特有蛋白 RBA1 识别病原体效应物来调节拟南芥细胞死亡

Marc T Nishimura, Ryan G Anderson, Karen A Cherkis, Terry F Law, Qingli L Liu, Mischa Machius, Zachary L Nimchuk, Li Yang, Eui-Hwan Chung, Farid El Kasmi, Michael Hyunh, Erin Osborne Nishimura, John E Sondek, Jeffery L Dangl

Structural analyses to identify selective inhibitors of glyceraldehyde 3-phosphate dehydrogenase-S, a sperm-specific glycolytic enzyme

通过结构分析鉴定精子特异性糖酵解酶甘油醛 3-磷酸脱氢酶-S 的选择性抑制剂

Polina V Danshina, Weidong Qu, Brenda R Temple, Rafael J Rojas, Michael J Miley, Mischa Machius, Laurie Betts, Deborah A O'Brien

Discovery of Mer specific tyrosine kinase inhibitors for the treatment and prevention of thrombosis

发现用于治疗和预防血栓形成的 Mer 特异性酪氨酸激酶抑制剂

Weihe Zhang, Andrew L McIver, Michael A Stashko, Deborah DeRyckere, Brian R Branchford, Debra Hunter, Dmitri Kireev, Michael J Miley, Jacqueline Norris-Drouin, Wendy M Stewart, Minjung Lee, Susan Sather, Yingqiu Zhou, Jorge A Di Paola, Mischa Machius, William P Janzen, H Shelton Earp, Douglas K Grah

Pseudo-cyclization through intramolecular hydrogen bond enables discovery of pyridine substituted pyrimidines as new Mer kinase inhibitors

通过分子内氢键进行伪环化,发现吡啶取代的嘧啶作为新的 Mer 激酶抑制剂

Weihe Zhang, Dehui Zhang, Michael A Stashko, Deborah DeRyckere, Debra Hunter, Dmitri Kireev, Michael J Miley, Christopher Cummings, Minjung Lee, Jacqueline Norris-Drouin, Wendy M Stewart, Susan Sather, Yingqiu Zhou, Gregory Kirkpatrick, Mischa Machius, William P Janzen, H Shelton Earp, Douglas K Gra

Structural determinants of RGS-RhoGEF signaling critical to Entamoeba histolytica pathogenesis

RGS-RhoGEF 信号的结构决定因素对溶组织内阿米巴发病机制至关重要

Dustin E Bosch, Adam J Kimple, Alyssa J Manning, Robin E Muller, Francis S Willard, Mischa Machius, Stephen L Rogers, David P Siderovski