日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A covalent inhibitor of the YAP-TEAD transcriptional complex identified by high-throughput screening

通过高通量筛选鉴定出 YAP-TEAD 转录复合物的共价抑制剂

Kayla Nutsch, Lirui Song, Emily Chen, Mitchell Hull, Arnab K Chatterjee, Jian Jeffery Chen, Michael J Bollong

High throughput screening for drugs that inhibit 3C-like protease in SARS-CoV-2

高通量筛选抑制 SARS-CoV-2 中 3C 样蛋白酶的药物

Emery Smith, Meredith E Davis-Gardner, Ruben D Garcia-Ordonez, Tu-Trinh Nguyen, Mitchell Hull, Emily Chen, Xuerong Yu, Thomas D Bannister, Pierre Baillargeon, Louis Scampavia, Patrick Griffin, Michael Farzan, Timothy P Spicer

Identification of potent small molecule inhibitors of SARS-CoV-2 entry

鉴定有效的 SARS-CoV-2 入侵小分子抑制剂

Sonia Mediouni, Huihui Mou, Yuka Otsuka, Joseph Anthony Jablonski, Robert Scott Adcock, Lalit Batra, Dong-Hoon Chung, Christopher Rood, Ian Mitchelle S de Vera, Ronald Rahaim Jr, Sultan Ullah, Xuerong Yu, Yulia A Getmanenko, Nicole M Kennedy, Chao Wang, Tu-Trinh Nguyen, Mitchell Hull, Emily Chen, Th

YAP-dependent proliferation by a small molecule targeting annexin A2

靶向膜联蛋白 A2 的小分子促进 YAP 依赖性增殖

Sophia Z Shalhout #, Peng-Yu Yang #, Edyta M Grzelak #, Kayla Nutsch, Sida Shao, Claudio Zambaldo, Jonathan Iaconelli, Lara Ibrahim, Caroline Stanton, Stormi R Chadwick, Emily Chen, Michael DeRan, Sijia Li, Mitchell Hull, Xu Wu, Arnab K Chatterjee, Weijun Shen, Fernando D Camargo, Peter G Schultz, M

Bispecific repurposed medicines targeting the viral and immunological arms of COVID-19

针对新冠病毒病毒和免疫系统的双特异性再利用药物

Martin A Redhead,C David Owen,Lennart Brewitz,Amelia H Collette,Petra Lukacik,Claire Strain-Damerell,Sean W Robinson,Patrick M Collins,Philipp Schäfer,Mark Swindells,Chris J Radoux,Iva Navratilova Hopkins,Daren Fearon,Alice Douangamath,Frank von Delft,Tika R Malla,Laura Vangeel,Thomas Vercruysse,Jan Thibaut,Pieter Leyssen,Tu-Trinh Nguyen,Mitchell Hull,Anthony Tumber,David J Hallett,Christopher J Schofield,David I Stuart,Andrew L Hopkins,Martin A Walsh

High-Throughput Screening for Drugs That Inhibit Papain-Like Protease in SARS-CoV-2

高通量筛选抑制 SARS-CoV-2 木瓜蛋白酶样蛋白酶的药物

Emery Smith, Meredith E Davis-Gardner, Ruben D Garcia-Ordonez, Tu-Trinh Nguyen, Mitchell Hull, Emily Chen, Pierre Baillargeon, Louis Scampavia, Timothy Strutzenberg, Patrick R Griffin, Michael Farzan, Timothy P Spicer

Selective BET bromodomain inhibition as an antifungal therapeutic strategy

选择性 BET 溴结构域抑制作为抗真菌治疗策略

Flore Mietton, Elena Ferri, Morgane Champleboux, Ninon Zala, Danièle Maubon, Yingsheng Zhou, Mike Harbut, Didier Spittler, Cécile Garnaud, Marie Courçon, Murielle Chauvel, Christophe d'Enfert, Boris A Kashemirov, Mitchell Hull, Muriel Cornet, Charles E McKenna, Jérôme Govin, Carlo Petosa