日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Agricultural innovations for sustainability? Diverse pathways and plural perspectives on rice seeds in Odisha, India

农业创新促进可持续发展?印度奥里萨邦水稻种子的多样化路径和多元视角

Arora, Saurabh; Narayanarao, Bhuvana; Mittal, Nimisha; Vadekkal, Rasheed Sulaiman

Discovery of Potent Antimalarial Type II Kinase Inhibitors with Selectivity over Human Kinases.

发现对人类激酶具有选择性的强效抗疟疾 II 型激酶抑制剂

Wang Lushun, Bohmer Monica J, Wang Jinhua, Nardella Flore, Calla Jaeson, Laureano De Souza Mariana, Schindler Kyra A, Montejo Lukas, Mittal Nimisha, Rocamora Frances, Treat Mayland, Charlton Jordan T, Tumwebaze Patrick K, Rosenthal Philip J, Cooper Roland A, Chakrabarti Ratna, Winzeler Elizabeth A, Chakrabarti Debopam, Gray Nathanael S

Exploration and characterization of the antimalarial activity of cyclopropyl carboxamides that target the mitochondrial protein, cytochrome b

探索和表征靶向线粒体蛋白细胞色素b的环丙基羧酰胺类化合物的抗疟活性

Awalt, Jon Kyle; Su, Wenyin; Nguyen, William; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Ramesh, Saishyam; Fairhurst, Kate J; Yeo, Tomas; Park, Heekuk; Uhlemann, Anne-Catrin; Chandra Maity, Bikash; De, Nirupam; Mukherjee, Partha; Chakraborty, Arnish; Churchyard, Alisje; Famodimu, Mufuliat T; Delves, Michael J; Baum, Jake; Mittal, Nimisha; Winzeler, Elizabeth A; Papenfuss, Anthony T; Chowdury, Mrittika; de Koning-Ward, Tania F; Maier, Alexander G; van Dooren, Giel G; Baud, Delphine; Brand, Stephen; Fidock, David A; Jackson, Paul F; Cowman, Alan F; Dans, Madeline G; Sleebs, Brad E

Fast-Killing Tyrosine Amide ((S)-SW228703) with Blood- and Liver-Stage Antimalarial Activity Associated with the Cyclic Amine Resistance Locus (PfCARL)

快速杀灭酪氨酸酰胺((S)-SW228703)具有血液期和肝脏期抗疟活性,与环胺抗性基因座(PfCARL)相关

Imlay, Leah S; Lawong, Aloysus K; Gahalawat, Suraksha; Kumar, Ashwani; Xing, Chao; Mittal, Nimisha; Wittlin, Sergio; Churchyard, Alisje; Niederstrasser, Hanspeter; Crespo-Fernandez, Benigno; Posner, Bruce A; Gamo, Francisco-Javier; Baum, Jake; Winzeler, Elizabeth A; Laleu, Benoît; Ready, Joseph M; Phillips, Margaret A

Design of proteasome inhibitors with oral efficacy in vivo against Plasmodium falciparum and selectivity over the human proteasome

设计对恶性疟原虫具有体内口服疗效且对人蛋白酶体具有选择性的蛋白酶体抑制剂

Xie, Stanley C; Metcalfe, Riley D; Mizutani, Hirotake; Puhalovich, Tanya; Hanssen, Eric; Morton, Craig J; Du, Yawei; Dogovski, Con; Huang, Shih-Chung; Ciavarri, Jeffrey; Hales, Paul; Griffin, Robert J; Cohen, Lawrence H; Chuang, Bei-Ching; Wittlin, Sergio; Deni, Ioanna; Yeo, Tomas; Ward, Kurt E; Barry, Daniel C; Liu, Boyin; Gillett, David L; Crespo-Fernandez, Benigno F; Ottilie, Sabine; Mittal, Nimisha; Churchyard, Alisje; Ferguson, Daniel; Aguiar, Anna Caroline C; Guido, Rafael V C; Baum, Jake; Hanson, Kirsten K; Winzeler, Elizabeth A; Gamo, Francisco-Javier; Fidock, David A; Baud, Delphine; Parker, Michael W; Brand, Stephen; Dick, Lawrence R; Griffin, Michael D W; Gould, Alexandra E; Tilley, Leann

Potent Antimalarials with Development Potential Identified by Structure-Guided Computational Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series

通过基于吡咯的二氢乳清酸脱氢酶抑制剂系列的结构导向计算优化,鉴定出具有开发潜力的强效抗疟药物

Palmer, Michael J; Deng, Xiaoyi; Watts, Shawn; Krilov, Goran; Gerasyuto, Aleksey; Kokkonda, Sreekanth; El Mazouni, Farah; White, John; White, Karen L; Striepen, Josefine; Bath, Jade; Schindler, Kyra A; Yeo, Tomas; Shackleford, David M; Mok, Sachel; Deni, Ioanna; Lawong, Aloysus; Huang, Ann; Chen, Gong; Wang, Wen; Jayaseelan, Jaya; Katneni, Kasiram; Patil, Rahul; Saunders, Jessica; Shahi, Shatrughan P; Chittimalla, Rajesh; Angulo-Barturen, Iñigo; Jiménez-Díaz, María Belén; Wittlin, Sergio; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Aguiar, Anna Caroline Campos; Guido, Rafael V C; Pereira, Dhelio B; Mittal, Nimisha; Winzeler, Elizabeth A; Tomchick, Diana R; Laleu, Benoît; Burrows, Jeremy N; Rathod, Pradipsinh K; Fidock, David A; Charman, Susan A; Phillips, Margaret A

The mitochondrial SIR2 related protein 2 (SIR2RP2) impacts Leishmania donovani growth and infectivity

线粒体SIR2相关蛋白2 (SIR2RP2) 影响杜氏利什曼原虫的生长和感染力。

Mittal, Nimisha; Muthuswami, Rohini; Madhubala, Rentala