日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

SARM1 activation induces reversible mitochondrial dysfunction and can be prevented in human neurons by antisense oligonucleotides.

SARM1 激活可导致可逆性线粒体功能障碍,而反义寡核苷酸可以预防人类神经元中的这种功能障碍

Loreto Andrea, Cramb Kaitlyn M L, McDermott Lucy A, Antoniou Christina, Cirilli Ilenia, Caiazza Maria Claudia, Merlini Elisa, Arthur-Farraj Peter, du Preez W Daniel, Mock Elliot D, Zhao Hien T, Bennett David L, Orsomando Giuseppe, Coleman Michael P, Wade-Martins Richard

Activity-Based Protein Profiling Identifies α-Ketoamides as Inhibitors for Phospholipase A2 Group XVI

基于活性的蛋白质谱分析鉴定出α-酮酰胺是磷脂酶A2第十六组的抑制剂

Zhou, Juan; Mock, Elliot D; Martella, Andrea; Kantae, Vasudev; Di, Xinyu; Burggraaff, Lindsey; Baggelaar, Marc P; Al-Ayed, Karol; Bakker, Alexander; Florea, Bogdan I; Grimm, Sebastian H; den Dulk, Hans; Li, Chun T; Mulder, Laura; Overkleeft, Herman S; Hankemeier, Thomas; van Westen, Gerard J P; van der Stelt, Mario

Activity-based protein profiling reveals off-target proteins of the FAAH inhibitor BIA 10-2474

基于活性的蛋白质谱分析揭示了FAAH抑制剂BIA 10-2474的脱靶蛋白

van Esbroeck, Annelot C M; Janssen, Antonius P A; Cognetta, Armand B 3rd; Ogasawara, Daisuke; Shpak, Guy; van der Kroeg, Mark; Kantae, Vasudev; Baggelaar, Marc P; de Vrij, Femke M S; Deng, Hui; Allarà, Marco; Fezza, Filomena; Lin, Zhanmin; van der Wel, Tom; Soethoudt, Marjolein; Mock, Elliot D; den Dulk, Hans; Baak, Ilse L; Florea, Bogdan I; Hendriks, Giel; De Petrocellis, Luciano; Overkleeft, Herman S; Hankemeier, Thomas; De Zeeuw, Chris I; Di Marzo, Vincenzo; Maccarrone, Mauro; Cravatt, Benjamin F; Kushner, Steven A; van der Stelt, Mario