Tetrahydropyrazolo[1,5-a]pyrimidine-3-carboxamide and N-benzyl-6',7'-dihydrospiro[piperidine-4,4'-thieno[3,2-c]pyran] analogues with bactericidal efficacy against Mycobacterium tuberculosis targeting MmpL3
四氢吡唑并[1,5-a]嘧啶-3-甲酰胺和N-苄基-6',7'-二氢螺[哌啶-4,4'-噻吩并[3,2-c]吡喃]类似物对结核分枝杆菌具有杀菌活性,靶向MmpL3
期刊:PLoS One
影响因子:2.6
doi:10.1371/journal.pone.0060933
Remuiñán, Modesto J; Pérez-Herrán, Esther; Rullás, Joaquín; Alemparte, Carlos; Martínez-Hoyos, María; Dow, David J; Afari, Johnson; Mehta, Nalini; Esquivias, Jorge; Jiménez, Elena; Ortega-Muro, Fátima; Fraile-Gabaldón, María Teresa; Spivey, Vickey L; Loman, Nicholas J; Pallen, Mark J; Constantinidou, Chrystala; Minick, Douglas J; Cacho, Mónica; Rebollo-López, María José; González, Carolina; Sousa, Verónica; Angulo-Barturen, Iñigo; Mendoza-Losana, Alfonso; Barros, David; Besra, Gurdyal S; Ballell, Lluís; Cammack, Nicholas