Discovery of potent BET bromodomain 1 stereoselective inhibitors using DNA-encoded chemical library selections
利用DNA编码化学库筛选发现强效BET溴结构域1立体选择性抑制剂
期刊:Proceedings of the National Academy of Sciences of the United States of America
影响因子:9.1
doi:10.1073/pnas.2122506119
Modukuri, Ram K; Yu, Zhifeng; Tan, Zhi; Ta, Hai Minh; Ucisik, Melek Nihan; Jin, Zhuang; Anglin, Justin L; Sharma, Kiran L; Nyshadham, Pranavanand; Li, Feng; Riehle, Kevin; Faver, John C; Duong, Kevin; Nagarajan, Sureshbabu; Simmons, Nicholas; Palmer, Stephen S; Teng, Mingxing; Young, Damian W; Yi, Joanna S; Kim, Choel; Matzuk, Martin M