日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The molecular basis of intrinsic resistance to azoles in Rhizopus arrhizus

根霉对唑类药物固有抗性的分子基础

Lackner, Michaela; Toepfer, Stephanie; Keniya, Mikhail V; Lax, Carlos; Nicolas, Francisco E; Garre, Victoriano; Müller, Christoph; Rosam, Katharina; Zenz, Lisa-Maria; Cesarini, Lucia; Binder, Ulrike; Tyndall, Joel D A; Monk, Brian C

Exploring Long Arm Amide-Linked Side Chains in the Design of Antifungal Azole Inhibitors of Sterol 14α-Demethylase (CYP51)

探索长臂酰胺连接侧链在甾醇14α-去甲基酶(CYP51)抗真菌唑类抑制剂设计中的应用

Alsulaimany, Marwa; Keniya, Mikhail V; Alanazi, Rehab S; N Ruma, Yasmeen; Hughes, Carwyn S; Jones, Arwyn T; Tyndall, Joel D A; Parker, Josie E; Monk, Brian C; Simons, Claire

Azole Combinations and Multi-Targeting Drugs That Synergistically Inhibit Candidozyma auris

唑类化合物和多靶点药物协同抑制耳念珠菌

Toepfer, Stephanie; Keniya, Mikhail V; Lackner, Michaela; Monk, Brian C

The Molecular Basis of the Intrinsic and Acquired Resistance to Azole Antifungals in Aspergillus fumigatus.

烟曲霉对唑类抗真菌药物固有耐药性和获得性耐药性的分子基础

Hosseini Parham, Keniya Mikhail V, Sagatova Alia A, Toepfer Stephanie, Müller Christoph, Tyndall Joel D A, Klinger Anette, Fleischer Edmond, Monk Brian C

Exploring Cryptococcus neoformans CYP51 and Its Cognate Reductase as a Drug Target

探索新型隐球菌CYP51及其同源还原酶作为药物靶点

Ruma, Yasmeen N; Keniya, Mikhail V; Monk, Brian C

Roles for Structural Biology in the Discovery of Drugs and Agrochemicals Targeting Sterol 14α-Demethylases

结构生物学在发现靶向甾醇14α-去甲基酶的药物和农用化学品中的作用

Monk, Brian C; Keniya, Mikhail V

Structural Insights into the Azole Resistance of the Candida albicans Darlington Strain Using Saccharomyces cerevisiae Lanosterol 14α-Demethylase as a Surrogate

利用酿酒酵母羊毛甾醇14α-去甲基酶作为替代物,深入了解白色念珠菌达林顿菌株的唑类耐药性

Graham, Danyon O; Wilson, Rajni K; Ruma, Yasmeen N; Keniya, Mikhail V; Tyndall, Joel D A; Monk, Brian C

Directed Mutational Strategies Reveal Drug Binding and Transport by the MDR Transporters of Candida albicans

定向突变策略揭示白色念珠菌多药耐药转运蛋白的药物结合和转运机制

Banerjee, Atanu; Pata, Jorgaq; Sharma, Suman; Monk, Brian C; Falson, Pierre; Prasad, Rajendra

Correction: Monk, B.C.; Keniya, M.V. Roles for Structural Biology in the Discovery of Drugs and Agrochemicals Targeting Sterol 14α-Demethylases. J. Fungi 2021, 7, 67

更正:Monk, BC; Keniya, MV. 结构生物学在发现靶向甾醇14α-去甲基酶的药物和农用化学品中的作用。J. Fungi 2021, 7, 67

Monk, Brian C; Keniya, Mikhail V

Highlighting membrane protein structure and function: A celebration of the Protein Data Bank

聚焦膜蛋白结构与功能:蛋白质数据库的盛会

Li, Fei; Egea, Pascal F; Vecchio, Alex J; Asial, Ignacio; Gupta, Meghna; Paulino, Joana; Bajaj, Ruchika; Dickinson, Miles Sasha; Ferguson-Miller, Shelagh; Monk, Brian C; Stroud, Robert M