日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

A FAN1 point mutation associated with accelerated Huntington's disease progression alters its PCNA-mediated assembly on DNA

与亨廷顿病进展加速相关的FAN1基因点突变会改变其在DNA上通过PCNA介导的组装。

Aretz, Jonas; Jeyasankar, Gayathri; Salerno-Kochan, Anna; Thomsen, Maren; Thieulin-Pardo, Gabriel; Haque, Tasir; Monteagudo, Edith; Felsenfeld, Dan; Finley, Michael; Vogt, Thomas F; Boudet, Julien; Prasad, Brinda C

Elucidation of multiple high-resolution states of human MutSβ by cryo-EM reveals interplay between ATP/ADP binding and heteroduplex DNA recognition.

通过冷冻电镜阐明人类 MutSβ 的多个高分辨率状态,揭示了 ATP/ADP 结合和异源双链 DNA 识别之间的相互作用

Lee Jung-Hoon, Thomsen Maren, Daub Herwin, Thieulin-Pardo Gabriel, Steinbacher Stefan, Sztyler Agnieszka, Dahiya Vinay, Neudegger Tobias, Dominguez Celia, Iyer Ravi R, Wilkinson Hilary A, Monteagudo Edith, Plotnikov Nikolay V, Felsenfeld Dan P, Haque Tasir S, Finley Michael, Boudet Julien, Vogt Thomas F, Prasad Brinda C

Personalized Metabolic Profile by Synergic Use of NMR and HRMS

利用核磁共振和高分辨率质谱协同作用构建个性化代谢谱

Petrella, Greta; Montesano, Camilla; Lentini, Sara; Ciufolini, Giorgia; Vanni, Domitilla; Speziale, Roberto; Salonia, Andrea; Montorsi, Francesco; Summa, Vincenzo; Vago, Riccardo; Orsatti, Laura; Monteagudo, Edith; Cicero, Daniel Oscar

5,6-Dihydroxypyrimidine Scaffold to Target HIV-1 Nucleocapsid Protein

5,6-二羟基嘧啶骨架靶向HIV-1核衣壳蛋白

Malancona, Savina; Mori, Mattia; Fezzardi, Paola; Santoriello, Marisabella; Basta, Andreina; Nibbio, Martina; Kovalenko, Lesia; Speziale, Roberto; Battista, Maria Rosaria; Cellucci, Antonella; Gennari, Nadia; Monteagudo, Edith; Di Marco, Annalise; Giannini, Alessia; Sharma, Rajhans; Pires, Manuel; Real, Eleonore; Zazzi, Maurizio; Dasso Lang, Maria Chiara; De Forni, Davide; Saladini, Francesco; Mely, Yves; Summa, Vincenzo; Harper, Steven; Botta, Maurizio

Improved Selective Class I HDAC and Novel Selective HDAC3 Inhibitors: Beyond Hydroxamic Acids and Benzamides

改良型选择性I类HDAC抑制剂和新型选择性HDAC3抑制剂:超越羟肟酸和苯甲酰胺

Bresciani, Alberto; Ontoria, Jesus M; Biancofiore, Ilaria; Cellucci, Antonella; Ciammaichella, Alina; Di Marco, Annalise; Ferrigno, Federica; Francone, Alessandra; Malancona, Savina; Monteagudo, Edith; Nizi, Emanuela; Pace, Paola; Ponzi, Simona; Rossetti, Ilaria; Veneziano, Maria; Summa, Vincenzo; Harper, Steven

Discovery of a Selective Series of Inhibitors of Plasmodium falciparum HDACs

发现一系列选择性抑制恶性疟原虫 HDAC 的抑制剂

Ontoria, Jesus M; Paonessa, Giacomo; Ponzi, Simona; Ferrigno, Federica; Nizi, Emanuela; Biancofiore, Ilaria; Malancona, Savina; Graziani, Rita; Roberts, David; Willis, Paul; Bresciani, Alberto; Gennari, Nadia; Cecchetti, Ottavia; Monteagudo, Edith; Orsale, Maria V; Veneziano, Maria; Di Marco, Annalise; Cellucci, Antonella; Laufer, Ralph; Altamura, Sergio; Summa, Vincenzo; Harper, Steven

Discovery and Characterization of Novel Anti-schistosomal Properties of the Anti-anginal Drug, Perhexiline and Its Impact on Schistosoma mansoni Male and Female Reproductive Systems

抗心绞痛药物哌克西林新型抗血吸虫特性的发现与表征及其对曼氏血吸虫雄性和雌性生殖系统的影响

Guidi, Alessandra; Lalli, Cristiana; Perlas, Emerald; Bolasco, Giulia; Nibbio, Martina; Monteagudo, Edith; Bresciani, Alberto; Ruberti, Giovina

MK-5172, a Selective Inhibitor of Hepatitis C Virus NS3/4a Protease with Broad Activity across Genotypes and Resistant Variants

MK-5172,一种选择性抑制丙型肝炎病毒NS3/4a蛋白酶的药物,对多种基因型和耐药变异株均具有广泛活性。

Draper, Michael P; Weir, S; Macone, A; Donatelli, J; Trieber, C A; Tanaka, S K; Levy, Stuart B; P, Shahul Hameed; Solapure, Suresh; Mukherjee, Kakoli; Nandi, Vrinda; Waterson, David; Shandil, Radha; Balganesh, Meenakshi; Sambandamurthy, Vasan K; Raichurkar, Anand Kumar; Deshpande, Abhijeet; Ghosh, Anirban; Awasthy, Disha; Shanbhag, Gajanan; Sheikh, Gulebahar; McMiken, Helen; Puttur, Jayashree; Reddy, Jitendar; Werngren, Jim; Read, Jon; Kumar, Mahesh; R, Manjunatha; Chinnapattu, Murugan; Madhavapeddi, Prashanti; Manjrekar, Praveena; Basu, Reetobrata; Gaonkar, Sheshagiri; Sharma, Sreevalli; Hoffner, Sven; Humnabadkar, Vaishali; Subbulakshmi, Venkita; Panduga, Vijender; Summa, Vincenzo; Ludmerer, Steven W; McCauley, John A; Fandozzi, Christine; Burlein, Christine; Claudio, Giuliano; Coleman, Paul J; DiMuzio, Jillian M; Ferrara, Marco; Filippo, Marcello Di; Gates, Adam T; Graham, Donald J; Harper, Steven; Hazuda, Daria J; Huang, Qian; McHale, Carolyn; Monteagudo, Edith; Pucci, Vincenzo; Rowley, Michael; Rudd, Michael T; Soriano, Aileen; Stahlhut, Mark W; Vacca, Joseph P; Olsen, David B; Liverton, Nigel J; Carroll, Steven S