日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Preclinical and Early Clinical Development of PTC596, a Novel Small-Molecule Tubulin-Binding Agent

新型小分子微管蛋白结合剂PTC596的临床前和早期临床开发

Jernigan, Finith; Branstrom, Arthur; Baird, John D; Cao, Liangxian; Dali, Mandar; Furia, Bansri; Kim, Min Jung; O'Keefe, Kylie; Kong, Ronald; Laskin, Oscar L; Colacino, Joseph M; Pykett, Mark; Mollin, Anna; Sheedy, Josephine; Dumble, Melissa; Moon, Young-Choon; Sheridan, Richard; Mühlethaler, Tobias; Spiegel, Robert J; Prota, Andrea E; Steinmetz, Michel O; Weetall, Marla

Targeted BMI1 inhibition impairs tumor growth in lung adenocarcinomas with low CEBPα expression

靶向抑制BMI1可抑制CEBPα低表达肺腺癌的肿瘤生长

Yong, Kol Jia; Basseres, Daniela S; Welner, Robert S; Zhang, Wen Cai; Yang, Henry; Yan, Benedict; Alberich-Jorda, Meritxell; Zhang, Junyan; de Figueiredo-Pontes, Lorena Lobo; Battelli, Chiara; Hetherington, Christopher J; Ye, Min; Zhang, Hong; Maroni, Giorgia; O'Brien, Karen; Magli, Maria Cristina; Borczuk, Alain C; Varticovski, Lyuba; Kocher, Olivier; Zhang, Pu; Moon, Young-Choon; Sydorenko, Nadiya; Cao, Liangxian; Davis, Thomas W; Thakkar, Bhavin M; Soo, Ross A; Iwama, Atsushi; Lim, Bing; Halmos, Balazs; Neuberg, Donna; Tenen, Daniel G; Levantini, Elena

BMI-1 Targeting Interferes with Patient-Derived Tumor-Initiating Cell Survival and Tumor Growth in Prostate Cancer.

BMI-1靶向治疗干扰前列腺癌患者来源的肿瘤起始细胞的存活和肿瘤生长

Bansal Nitu, Bartucci Monica, Yusuff Shamila, Davis Stephani, Flaherty Kathleen, Huselid Eric, Patrizii Michele, Jones Daniel, Cao Liangxian, Sydorenko Nadiya, Moon Young-Choon, Zhong Hua, Medina Daniel J, Kerrigan John, Stein Mark N, Kim Isaac Y, Davis Thomas W, DiPaola Robert S, Bertino Joseph R, Sabaawy Hatem E