日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of KLHL12 Ligands Using Fragment-Based Methods

利用基于片段的方法鉴定KLHL12配体

Waterson, Alex G; Vadukoot, Anish; Jana, Somnath; Cui, Jianwen; Luong, Kelvin; Rietz, Tyson A; Madrigal-Carrillo, Ezequiel Alejandro; Lehmann, Brian D; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Petros, Zoe A; Scaggs, William Rush; Chacon Simon, Selena; Vekariya, Rakesh H; Kim, Kwangho; Thangaraj, Manikandan; Christov, Plamen P; South, Taylor M; Sai, Jiqing; Thiruvaipati, Anusha; Schmidt, Charles R; Eells, Rebecca; Moore, William J; Olejniczak, Edward T; Phan, Jason; Fesik, Stephen W

Expanded profiling of WD repeat domain 5 inhibitors reveals actionable strategies for the treatment of hematologic malignancies

对WD重复结构域5抑制剂的扩展分析揭示了治疗血液系统恶性肿瘤的可行策略

Meyer, Christian T; Smith, Brianna N; Wang, Jing; Teuscher, Kevin B; Grieb, Brian C; Howard, Gregory C; Silver, Alexander J; Lorey, Shelly L; Stott, Gordon M; Moore, William J; Lee, Taekyu; Savona, Michael R; Weissmiller, April M; Liu, Qi; Quaranta, Vito; Fesik, Stephen W; Tansey, William P

Structure-based discovery of potent WD repeat domain 5 inhibitors that demonstrate efficacy and safety in preclinical animal models

基于结构的高效WD重复结构域5抑制剂的发现,在临床前动物模型中证实了其疗效和安全性。

Teuscher, Kevin B; Chowdhury, Somenath; Meyers, Kenneth M; Tian, Jianhua; Sai, Jiqing; Van Meveren, Mayme; South, Taylor M; Sensintaffar, John L; Rietz, Tyson A; Goswami, Soumita; Wang, Jing; Grieb, Brian C; Lorey, Shelly L; Howard, Gregory C; Liu, Qi; Moore, William J; Stott, Gordon M; Tansey, William P; Lee, Taekyu; Fesik, Stephen W

Structure-Based Discovery of Potent, Orally Bioavailable Benzoxazepinone-Based WD Repeat Domain 5 Inhibitors

基于结构的高效、口服生物利用度高的苯并唑酮类WD重复结构域5抑制剂的发现

Teuscher, Kevin B; Mills, Jonathan J; Tian, Jianhua; Han, Changho; Meyers, Kenneth M; Sai, Jiqing; South, Taylor M; Crow, Mackenzie M; Van Meveren, Mayme; Sensintaffar, John L; Zhao, Bin; Amporndanai, Kangsa; Moore, William J; Stott, Gordon M; Tansey, William P; Lee, Taekyu; Fesik, Stephen W

1109. A multicenter, observational study to compare the effectiveness of Ceftazidime-Avibactam versus Ceftolozane-Tazobactam for multidrug-resistant Pseudomonas aeruginosa infections in the United States (CACTUS)

1109. 一项多中心观察性研究,比较头孢他啶-阿维巴坦与头孢洛扎-他唑巴坦治疗美国多重耐药铜绿假单胞菌感染的疗效(CACTUS)

Boyer, Edward W; Wines, James D Jr; Shields, Ryan K; Abbo, Lilian M; Ackley, Renee; Aitken, Samuel L; Albrecht, Benjamin; Babiker, Ahmed; Cifuentes, Renzo; Claeys, Kimberly C; DeSear, Kathryn; Gallagher, Jason C; Gregory, Eric; Heil, Emily L; Hickey, Carissa; Klatt, Megan; Kline, Ellen G; Kubat, Ryan C; Kufel, Wesley D; Hyoung Lee, Jae; Lim, Ahmi; Lingg, Theresa; MacDougall, Conan; Mathers, Amy; McCreary, Erin K; Moore, William J; Olson, Shannon; Oxer, Jessica; Pearson, Jeffrey C; Pham, Christine; Polk, Christopher; Satlin, Michael J; Satola, Sarah W; Shah, Sunish; Solanki, Yash B; Tamma, Pranita; Vega, Ana; Veena, Venugopalan; Veve, Michael; Wangchinda, Walaiporn; Witt, Lucy S; Wu, Janet; Pogue, jason M

Real-World Experience of Bamlanivimab for Coronavirus Disease 2019 (COVID-19): A Case-Control Study

巴姆拉尼维单抗治疗2019冠状病毒病(COVID-19)的真实世界经验:一项病例对照研究

Kumar, Rebecca N; Wu, En-Ling; Stosor, Valentina; Moore, William J; Achenbach, Chad; Ison, Michael G; Angarone, Michael P

Reply to Lapadula et al

回复 Lapadula 等人

Kumar, Rebecca N; Wu, En-Ling; Stosor, Valentina; Moore, William J; Achenbach, Chad; Ison, Michael G; Angarone, Michael P

180. Impact of a two-step diagnostic bundle on hospital-onset Clostridioides difficile infection rates and treatment across a large health system

180. 两步诊断方案对大型医疗系统中医院获得性艰难梭菌感染率和治疗的影响

Perlin, Mark William; Polisetty, Radhika S; Hoff, Brian M; Moore, William J; Postelnick, Michael; Wang, Sheila K; Zembower, Teresa; Chao, Qi; Malczynski, Michael; Barajas, Grace; Silkaitis, Christina; Salim, Asra; Borkowski, Jaime; Shah, Rishita; Quinn, Andrea; Johnicker, Kyle; Liang, Charlene; Chang, Stephanie; Sutton, Sarah H

Early Multicenter Experience With Imipenem-Cilastatin-Relebactam for Multidrug-Resistant Gram-Negative Infections

亚胺培南-西司他丁-瑞巴坦治疗多重耐药革兰氏阴性菌感染的早期多中心经验

Rebold, Nicholas; Morrisette, Taylor; Lagnf, Abdalhamid M; Alosaimy, Sara; Holger, Dana; Barber, Katie; Justo, Julie Ann; Antosz, Kayla; Carlson, Travis J; Frens, Jeremy J; Biagi, Mark; Kufel, Wesley D; Moore, William J; Mercuro, Nicholas; Raux, Brian R; Rybak, Michael J

Optimization of ether and aniline based inhibitors of lactate dehydrogenase

乳酸脱氢酶醚类和苯胺类抑制剂的优化

Christov, Plamen P; Kim, Kwangho; Jana, Somnath; Romaine, Ian M; Rai, Ganesha; Mott, Bryan T; Allweil, Alexander A; Lamers, Alexander; Brimacombe, Kyle R; Urban, Daniel J; Lee, Tobie D; Hu, Xin; Lukacs, Christine M; Davies, Douglas R; Jadhav, Ajit; Hall, Matthew D; Green, Neal; Moore, William J; Stott, Gordon M; Flint, Andrew J; Maloney, David J; Sulikowski, Gary A; Waterson, Alex G